SCHEMBL4056076

SCHEMBL4056076

CC(C)[C@@H](NCCCNC(=O)OC(C)(C)C)c1nc2c(Cl)cnn2c(=O)n1Cc1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 1/20 0.40
STK17B O94768 1/20 0.39
STK17A Q9UEE5 1/20 0.39
SIGMAR1 Q99720 2/20 0.37
CYP3A4 P08684 1/20 0.37
TLR7 Q9NYK1 5/20 0.36
BRD4 O60885 2/20 0.36
IL6 P05231 1/20 0.36
P2RX7 Q99572 1/20 0.36
SCD O00767 1/20 0.35
PDE1B Q01064 1/20 0.35
GNRHR P30968 1/20 0.35
NPSR1 Q6W5P4 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4056075 1.00 KIF11 (0.40) KIF11STK17BSTK17ASIGMAR1CYP3A4
SCHEMBL4004013 0.89 KIF11 (0.43) KIF11STK17BSTK17ASIGMAR1CYP3A4
SCHEMBL4050591 0.87 KIF11 (0.41) KIF11STK17BSTK17ASIGMAR1BRD4
SCHEMBL4055834 0.87 KIF11 (0.41) KIF11STK17BSTK17ASIGMAR1BRD4
SCHEMBL4049089 0.86 KIF11 (0.39) KIF11SIGMAR1TLR7BRD4PDE1B
SCHEMBL4056718 0.85 KIF11 (0.41) KIF11TLR7BRD4NPSR1L3MBTL1
SCHEMBL4056720 0.85 KIF11 (0.41) KIF11TLR7BRD4NPSR1L3MBTL1
SCHEMBL13963456 0.82 SIGMAR1 (0.42) KIF11SIGMAR1CYP3A4BRD4GNRHR
SCHEMBL4054974 0.82 KIF11 (0.39) KIF11BRD4P2RX7GNRHR
SCHEMBL4054984 0.82 KIF11 (0.39) KIF11BRD4P2RX7GNRHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2070932-A1 Pyrazolotriazines 4SC AG (DE) 2009-06-17 EP disclosed