SCHEMBL4056677

SCHEMBL4056677

Cc1ccc(CO)cc1[NH]

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 1/20 0.43
S1PR1 P21453 3/20 0.37
PRSS1 P07477 2/20 0.35
PRSS2 P07478 2/20 0.35
PRSS3 P35030 2/20 0.35
ESR1 P03372 1/20 0.35
ESR2 Q92731 1/20 0.35
CYP4F2 P78329 1/20 0.34
CYP4A11 Q02928 1/20 0.34
RECQL P46063 1/20 0.33
TSHR P16473 1/20 0.33
MAOA P21397 1/20 0.33
DYRK1A Q13627 1/20 0.33
ENPP2 Q13822 1/20 0.33
GRM2 Q14416 1/20 0.33
CA12 O43570 1/20 0.32
CA2 P00918 1/20 0.32
CA3 P07451 1/20 0.32
CA4 P22748 1/20 0.32
CA6 P23280 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4134649 0.82 ESR1 (0.40) HSD17B10S1PR1PRSS1PRSS2PRSS3
SCHEMBL93048 0.78 S1PR1 (0.47) HSD17B10S1PR1PRSS1PRSS2PRSS3
SCHEMBL148755 0.76 SHBG (0.48) HSD17B10S1PR1ESR1ESR2CYP4F2
SCHEMBL29741490 0.76 SHBG (0.48) HSD17B10S1PR1ESR1ESR2CYP4F2
SCHEMBL1950124 0.74 TSHR (0.48) HSD17B10ESR1ESR2RECQLTSHR
SCHEMBL31371255 0.74 TSHR (0.48) HSD17B10ESR1ESR2RECQLTSHR
Phosphonic Acid SCHEMBL4098634 0.74 S1PR1 (0.41) HSD17B10S1PR1PRSS1PRSS2PRSS3
SCHEMBL92958 0.73 S1PR1 (0.51) HSD17B10S1PR1RECQLTTR
SCHEMBL2208303 0.73 S1PR1 (0.41) HSD17B10S1PR1ESR1ESR2CYP4F2
SCHEMBL1467659 0.73 HPGD (0.42) HSD17B10S1PR1ESR1ESR2CYP4F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7547713-B2 O-pyridinequinone derivatives, the composition containing the derivatives, the process for preparation of the derivatives and the use of the derivatives GU LIANQUAN 2009-06-16 US claimed
US-20060111405-A1 O-pyridinequinone derivatives, the composition containing the derivatives, the process for preparation of the derivatives and the use of the derivatives GU LIANQUAN 2006-05-25 US claimed
US-7547713-B2 O-pyridinequinone derivatives, the composition containing the derivatives, the process for preparation of the derivatives and the use of the derivatives GU LIANQUAN 2009-06-16 US disclosed
US-20060111405-A1 O-pyridinequinone derivatives, the composition containing the derivatives, the process for preparation of the derivatives and the use of the derivatives GU LIANQUAN 2006-05-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060111405-A1 O-pyridinequinone derivatives, the composition containing the derivatives, the process for preparation of the derivatives and the use of the derivatives PTGS2, PTGES2, PTGES HSD17B10 1258/4885S1PR1 4147/4885PRSS1 3144/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.