Tramadol

Tramadol

SCHEMBL405855

COc1cccc(C2(O)CCCCC2CN(C)C)c1.Cl

nearest known ligand 0.98

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

OPRM1

The experimentally established mechanism targets of Tramadol. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
OPRM1 known ✓ P35372 11/20 0.98
SLC6A2 P23975 13/20 0.98
SLC6A4 P31645 13/20 0.98
OPRD1 P41143 6/20 0.98
OPRK1 P41145 4/20 0.98
SLC22A1 O15245 3/20 0.98
MEN1 O00255 2/20 0.98
KMT2A Q03164 2/20 0.98
CHRM2 P08172 1/20 0.98
CHRM1 P11229 1/20 0.98

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
(R,R)-Tramadol SCHEMBL29625842 1.00 SLC6A2 (0.98) SLC6A2SLC6A4OPRM1OPRD1OPRK1
(R,R)-Tramadol SCHEMBL429520 1.00 SLC6A2 (0.98) SLC6A2SLC6A4OPRM1OPRD1OPRK1
(R,R)-Tramadol SCHEMBL405854 1.00 SLC6A2 (0.98) SLC6A2SLC6A4OPRM1OPRD1OPRK1
(R,R)-Tramadol SCHEMBL41748 1.00 SLC6A2 (0.98) SLC6A2SLC6A4OPRM1OPRD1OPRK1
(R,R)-Tramadol SCHEMBL7141021 1.00 SLC6A2 (0.98) SLC6A2SLC6A4OPRM1OPRD1OPRK1
(R,R)-Tramadol SCHEMBL1377516 1.00 SLC6A2 (0.98) SLC6A2SLC6A4OPRM1OPRD1OPRK1
(R,R)-Tramadol SCHEMBL405853 1.00 SLC6A2 (0.98) SLC6A2SLC6A4OPRM1OPRD1OPRK1
(R,R)-Tramadol SCHEMBL7137387 1.00 SLC6A2 (0.98) SLC6A2SLC6A4OPRM1OPRD1OPRK1
Tramadol SCHEMBL6052999 1.00 SLC6A2 (0.98) SLC6A2SLC6A4OPRM1OPRD1OPRK1
(R,R)-Tramadol SCHEMBL6543502 1.00 SLC6A2 (0.98) SLC6A2SLC6A4OPRM1OPRD1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 268 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240282425-A1 AUTHENTICATION METHODS AND SYSTEMS FOR DISPENSED PRESCRIPTIONS LOW GORDON KEITH (US) 2024-08-22 US claimed
CN-118127137-A Method for changing relative amplification speeds of different nucleic acid targets through pre-PCR 浙江自贸区锐赛生物医药科技有限公司 2024-06-04 CN claimed
CN-117965705-A Method for changing relative PCR amplification speed of different nucleic acid targets 上海锐赛循益生物技术有限公司 2024-05-03 CN claimed
WO-2003078380-A2 PROCESS FOR PREPARING TRAMADOL HYDROCHLORIDE AND/OR TRAMADOL MOMOHYDRATE JUBILANT ORGANOSYS LTD (GB) 2003-09-25 WO claimed
EP-1346978-A1 Process for preparing tramadol hydrochloride and/or tramadol monohydrate Jubilant Organosys Limited (IN) 2003-09-24 EP claimed
EP-0831082-B1 Process for the purification of (RR-SS)-2-dimethylaminomethyl-1-(3-methoxyphenyl)cyclohexanol hydrochloride CHEMAGIS LTD (IL) 2002-06-05 EP claimed
EP-0778262-B1 Process for the purification of (RR-SS)-2-dimethyl-aminomethyl-1-(3-methoxyphenyl)cyclohexanol and its salts CHEMAGIS LTD (IL) 2001-01-24 EP claimed
US-5877351-A REACTION WITH HYDROGEN BROMIDE WYCKOFF CHEMICAL COMPANY, INC. (US) 1999-03-02 US claimed
US-5874620-A ADDING AN ELECTROPHIOLIC REAGENT TO A MIXTURE OF (RR,SS)-TRAMADOL HYDROCHLORIDE AND ITS (RS,SR) GEOMETRICAL ISOMER; REGIOSELECTIVE REACTION WITH THE HYDROXYL GROUP OF THE RS,SR-TRAMADOL LEAVING PURE (RR,SS) ISOMER CHEMAGIS, LTD. (IL) 1999-02-23 US claimed
EP-0831082-A1 Process for the purification of (RR-SS)-2-dimethylaminomethyl-1-(3-methoxyphenyl)cyclohexanol hydrochloride Chemagis Ltd. (IL) 1998-03-25 EP claimed
US-5672755-A Process for the purification of (RR-SS)-2-dimethyl-aminomethyl-1-(3-methoxyphenyl)cyclohexanol and its salts CHEMAGIS LTD. (IL) 1997-09-30 US claimed
US-5414129-A Process for the purification of 2-[(dimethylamino)methyl]-1-(3-methoxyphenyl)cyclohexanol and its salts CHEMAGIS, LTD. (IL) 1995-05-09 US claimed
EP-4744652-A2 A METHOD OF FORMING A COMPOSITION COMPRISING A PROBIOTIC MICRO-ENCAPSULATED IN A DENATURED PLANT PROTEIN MATRIX Anabio Technologies Limited (IE) 2026-05-20 EP disclosed
US-12616661-B2 Composition for type II diabetics and for use in providing sustained energy release over time TEAGASC—The Agriculture and Food Development Authority (IE) 2026-05-05 US disclosed
EP-3972581-B1 PREBIOTIC COMPOSITIONS EVONIK OPERATIONS GMBH (DE) 2026-03-25 EP disclosed
US-12582647-B2 Systems and methods for treating an opioid-induced adverse pharmacodynamic response PURDUE PHARMA L.P. (US) 2026-03-24 US disclosed
US-5672755-A Process for the purification of (RR-SS)-2-dimethyl-aminomethyl-1-(3-methoxyphenyl)cyclohexanol and its salts CHEMAGIS LTD. (IL) 1997-09-30 US disclosed
EP-0778262-A2 Process for the purification of (RR-SS)-2-dimethyl-aminomethyl-1-(3-methoxyphenyl)cyclohexanol and its salts Chemagis Ltd. (IL) 1997-06-11 EP disclosed
US-5414129-A Process for the purification of 2-[(dimethylamino)methyl]-1-(3-methoxyphenyl)cyclohexanol and its salts CHEMAGIS, LTD. (IL) 1995-05-09 US disclosed
US-5414129-A Process for the purification of 2-[(dimethylamino)methyl]-1-(3-methoxyphenyl)cyclohexanol and its salts CHEMAGIS, LTD. (IL) 1995-05-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12582647-B2 Systems and methods for treating an opioid-induced adverse pharmacodynamic response OPRM1, OPRK1, OPRD1 OPRM1 1/4885SLC6A2 10/4885SLC6A4 14/4885
US-12616661-B2 Composition for type II diabetics and for use in providing sustained energy release over time GIPR, GLP1R, GPR119 OPRM1 3095/4885SLC6A2 2391/4885SLC6A4 2410/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.