SCHEMBL4062829

SCHEMBL4062829

O=CC(Br)c1cccc(I)c1

nearest known ligand 0.34

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 3/20 0.33
CYP3A4 P08684 2/20 0.33
CYP2D6 P10635 2/20 0.33
SLC6A2 P23975 2/20 0.33
SLC6A4 P31645 2/20 0.33
KCNH2 Q12809 2/20 0.33
FAAH O00519 1/20 0.32
MGLL Q99685 1/20 0.32
APP P05067 1/20 0.32
ERN1 O75460 1/20 0.31
TACR1 P25103 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5704333 0.82 CYP3A4 (0.34) SLC6A3CYP3A4CYP2D6SLC6A2SLC6A4
SCHEMBL540882 0.78 ALDH1A1 (0.47) SLC6A3CYP3A4CYP2D6SLC6A2SLC6A4
SCHEMBL21495049 0.78 ALDH1A1 (0.47) SLC6A3CYP3A4CYP2D6SLC6A2SLC6A4
SCHEMBL28420 0.76 SLC6A3 (0.37) SLC6A3CYP3A4CYP2D6SLC6A2SLC6A4
SCHEMBL2631570 0.76 TACR1 (0.36) SLC6A3CYP3A4CYP2D6SLC6A2SLC6A4
SCHEMBL16794983 0.76 FAAH (0.36) SLC6A3CYP3A4CYP2D6SLC6A2SLC6A4
SCHEMBL1701121 0.76 ADRB1 (0.43) SLC6A3CYP3A4
SCHEMBL169020 0.76 ACP3 (0.43)
SCHEMBL167914 0.76 HDAC4 (0.44) CYP3A4CYP2D6
SCHEMBL4960285 0.76 ACP3 (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015088564-A1 P2X4 RECEPTOR MODULATING COMPOUNDS SUNOVION PHARMACEUTICALS INC. (US) 2015-06-18 WO disclosed
WO-2015088565-A1 P2X4 RECEPTOR MODULATING COMPOUNDS AND METHODS OF USE THEREOF SUNOVION PHARMACEUTICALS INC. (US) 2015-06-18 WO disclosed
WO-2009123753-A1 INHIBITION OF BACTERIAL BIOFILMS WITH IMIDAZOLE-PHENYL DERIVATIVES NORTH CAROLINA STATE UNIVERSITY (US) 2009-10-08 WO disclosed