SCHEMBL4066711

SCHEMBL4066711

CCOC(=O)C1OC=C(c2cccc(CC(C)N(C)C(=O)OC(C)(C)C)c2)O1

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ACHE P22303 6/20 0.35
BCHE P06276 4/20 0.35
NFKB1 P19838 1/20 0.33
NFKB2 Q00653 1/20 0.33
RELA Q04206 1/20 0.33
CTSB P07858 1/20 0.33
CTSS P25774 1/20 0.33
CTSK P43235 1/20 0.33
PPARG P37231 10/20 0.32
PPARA Q07869 7/20 0.32
MAOA P21397 1/20 0.32
MAOB P27338 1/20 0.32
SLC7A5 Q01650 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4068940 0.90 NFKB1 (0.33) NFKB1NFKB2RELACTSBCTSS
SCHEMBL4065537 0.89 ACHE (0.39) ACHEBCHECTSBCTSSCTSK
SCHEMBL4063479 0.83 CTSS (0.43) CTSBCTSSCTSK
SCHEMBL4058035 0.80 CTSS (0.36) CTSBCTSSCTSKPPARGPPARA
SCHEMBL4066701 0.79 CYP4F2 (0.35) ACHEBCHENFKB1NFKB2RELA
SCHEMBL13210973 0.71 ACHE (0.45) ACHEBCHECTSBCTSSCTSK
SCHEMBL12050814 0.70 BCHE (0.53) ACHEBCHECTSBCTSSCTSK
SCHEMBL4068936 0.69 CYP4F2 (0.34) NFKB1NFKB2RELA
SCHEMBL13748626 0.69 CYP4F2 (0.34) NFKB1NFKB2RELA
SCHEMBL4065540 0.68 BCHE (0.36) ACHEBCHESLC7A5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7569676-B2 Ecstasy-class derivatives, immunogens, and antibodies and their use in detecting ecstasy-class drugs ROCHE DIAGNOSTICS OPERATIONS, INC. (US) 2009-08-04 US disclosed
EP-1498415-B1 Ecstasy-class derivatives, immunogens, and antibodies and their use in detecting ecstasy-class drugs ROCHE DIAGNOSTICS GMBH (DE) 2007-06-27 EP disclosed
US-7060847-B2 Ecstasy-class derivatives, immunogens, and antibodies and their use in detecting ecstasy-class drugs ROCHE DIAGNOSTICS OPERATIONS, INC. (US) 2006-06-13 US disclosed
US-20050153439-A1 Ecstasy-class derivatives, immunogens, and antibodies and their use in detecting ecstasy-class drugs GHOSHAL MITALI (US) 2005-07-14 US disclosed
US-20050014210-A1 Ecstasy-class derivatives, immunogens, and antibodies and their use in detecting ecstasy-class drugs ROCHE DIAGNOSTICS CORPORATION 2005-01-20 US disclosed
EP-1498415-A1 Ecstasy-class derivatives, immunogens, and antibodies and their use in detecting ecstasy-class drugs Roche Diagnostics GmbH (DE) 2005-01-19 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050014210-A1 Ecstasy-class derivatives, immunogens, and antibodies and their use in detecting ecstasy-class drugs DRD3, SLC6A3, DRD2 ACHE 130/4885BCHE 163/4885NFKB1 4552/4885
US-20050153439-A1 Ecstasy-class derivatives, immunogens, and antibodies and their use in detecting ecstasy-class drugs DRD3, SLC6A3, DRD2 ACHE 130/4885BCHE 163/4885NFKB1 4552/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.