SCHEMBL4068455

SCHEMBL4068455

CC(C)(C)OC(=O)N1CCN(C(C)(C)CN2CCCC2=O)CC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.42
MEN1 O00255 2/20 0.42
DDB1 Q16531 1/20 0.41
CRBN Q96SW2 1/20 0.41
USP2 O75604 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
MAPT P10636 2/20 0.39
PER2 O15055 1/20 0.38
HPGD P15428 1/20 0.38
TSHR P16473 1/20 0.38
ALDH1A1 P00352 2/20 0.38
DTYMK P23919 1/20 0.37
GPR119 Q8TDV5 1/20 0.37
CHRM2 P08172 1/20 0.37
CHRM4 P08173 1/20 0.37
CHRM1 P11229 1/20 0.37
CHRM3 P20309 1/20 0.37
NPC1 O15118 1/20 0.37
MAPK1 P28482 1/20 0.37
HTT P42858 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4206491 0.81 DTYMK (0.49) KMT2AMEN1DDB1CRBNUSP2
SCHEMBL16365258 0.80 ADRA1D (0.48) KMT2AMEN1DDB1CRBNUSP2
SCHEMBL189570 0.76 FPR2 (0.51) DDB1CRBNSMN1; SMN2MAPTHPGD
SCHEMBL8892804 0.76 KDM4E (0.55) SMN1; SMN2HPGDTSHRALDH1A1GPR119
SCHEMBL6778385 0.75 DTYMK (0.51) KMT2AMEN1DDB1CRBNUSP2
SCHEMBL1780574 0.74 USP2 (0.51) KMT2AMEN1USP2SMN1; SMN2MAPT
SCHEMBL1088328 0.74 USP2 (0.51) KMT2AMEN1DDB1CRBNUSP2
SCHEMBL29056036 0.73 FPR2 (0.50) MAPTHPGDGPR119NPC1RAB9A
SCHEMBL26129542 0.73 NR1H2 (0.44) KMT2AMEN1DDB1CRBNMAPT
SCHEMBL14585899 0.72 PLA2G7 (0.46) GPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2032582-A1 PYRIMIDINE DERIVATIVES AS PI3K INHIBITORS F.HOFFMANN-LA ROCHE AG (CH) 2009-03-11 EP disclosed
WO-2007122410-A1 PYRIMIDINE DERIVATIVES AS PI3K INHIBITORS F.HOFFMANN-LA ROCHE AG (CH) 2007-11-01 WO disclosed