SCHEMBL4068787

SCHEMBL4068787

CCNC(=O)Oc1cnc2c(c1)ncn2-c1ccc(OCc2ccc(OC(F)(F)F)cc2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 2/20 0.40
CYP19A1 P11511 1/20 0.40
CYP11B1 P15538 1/20 0.40
CYP11B2 P19099 1/20 0.40
PPARD Q03181 6/20 0.39
PPARA Q07869 6/20 0.39
PPARG P37231 4/20 0.39
GRM5 P41594 1/20 0.38
MAOB P27338 1/20 0.38
ADRB2 P07550 1/20 0.38
HPGD P15428 5/20 0.38
PDE2A O00408 1/20 0.38
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 2/20 0.38
MMP1 P03956 1/20 0.38
MMP2 P08253 1/20 0.38
MMP9 P14780 1/20 0.38
MMP14 P50281 1/20 0.38
ADAM17 P78536 1/20 0.38
CYP1A2 P05177 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4072391 0.92 MRGPRX4 (0.40) MRGPRX4CYP19A1CYP11B1CYP11B2GRM5
SCHEMBL4069211 0.91 MRGPRX4 (0.41) MRGPRX4CYP19A1CYP11B1CYP11B2PPARD
SCHEMBL4064790 0.90 MRGPRX4 (0.39) MRGPRX4CYP19A1CYP11B1CYP11B2PPARD
SCHEMBL4072173 0.89 ATM (0.40) MRGPRX4CYP19A1CYP11B1CYP11B2PPARD
SCHEMBL2961360 0.87 HPGD (0.44) MRGPRX4CYP19A1CYP11B1CYP11B2MAOB
SCHEMBL4061701 0.86 SMN1; SMN2 (0.44) CYP19A1CYP11B1CYP11B2ADRB2ALDH1A1
SCHEMBL4069255 0.86 MCHR1 (0.42) CYP19A1CYP11B1CYP11B2HPGDALDH1A1
SCHEMBL4065692 0.85 KDR (0.43) HPGDALDH1A1
SCHEMBL4066271 0.85 SLC6A5 (0.38) PPARDPPARAPPARGHPGDALDH1A1
SCHEMBL4061393 0.84 EPHX2 (0.44) GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1658289-B1 3-SUBSTITUTED IMIDAZOPYRIDINE-DERIVATIVES AS C-KIT INHIBITORS OSI PHARM INC (US) 2009-03-18 EP claimed