SCHEMBL4068903

SCHEMBL4068903

Cc1ccccc1C(=O)Nc1ccc(N(C)C2CCCCC2)nc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.51
L3MBTL1 Q9Y468 2/20 0.50
CYP1A2 P05177 1/20 0.49
TRPV1 Q8NER1 1/20 0.48
S1PR1 P21453 4/20 0.48
CRACR2A Q9BSW2 1/20 0.48
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
SMN1; SMN2 Q16637 3/20 0.47
RAB9A P51151 3/20 0.47
MAPT P10636 3/20 0.47
ALDH1A1 P00352 2/20 0.47
GAA P10253 2/20 0.47
MAPK1 P28482 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
PIK3CA P42336 1/20 0.46
MTOR P42345 1/20 0.46
HPGD P15428 1/20 0.46
KIT P10721 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4069506 0.88 SMN1; SMN2 (0.54) NPC1L3MBTL1TRPV1S1PR1MEN1
SCHEMBL4072949 0.88 S1PR1 (0.49) TRPV1S1PR1PIK3CAMTORHPGD
SCHEMBL4063941 0.80 S1PR1 (0.51) NPC1TRPV1S1PR1SMN1; SMN2RAB9A
SCHEMBL4064076 0.78 MEN1 (0.58) NPC1L3MBTL1CYP1A2TRPV1S1PR1
SCHEMBL4063306 0.76 L3MBTL1 (0.51) NPC1L3MBTL1CYP1A2S1PR1CRACR2A
SCHEMBL30010142 0.76 TRPV1 (0.55) NPC1L3MBTL1CYP1A2TRPV1SMN1; SMN2
SCHEMBL846037 0.74 TRPV1 (0.80) NPC1TRPV1SMN1; SMN2RAB9AALDH1A1
SCHEMBL25143492 0.74 HPGD (0.63) NPC1L3MBTL1CYP1A2SMN1; SMN2RAB9A
SCHEMBL31665584 0.74 HPGD (0.63) NPC1L3MBTL1CYP1A2SMN1; SMN2RAB9A
SCHEMBL4063294 0.73 MEN1 (0.53) NPC1L3MBTL1CYP1A2S1PR1CRACR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1028945-B9 SUBSTITUTED PYRIDINE COMPOUNDS AS ANTI-INFLAMMATORY AGENTS AMGEN INC (US) 2009-02-18 EP disclosed
EP-1028945-B1 SUBSTITUTED PYRIDINE COMPOUNDS AS ANTI-INFLAMMATORY AGENTS AMGEN INC (US) 2007-07-11 EP disclosed