SCHEMBL4073045

SCHEMBL4073045

CP(=O)(Cl)Oc1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SRC P12931 1/20 0.54
L3MBTL1 Q9Y468 2/20 0.52
TDP1 Q9NUW8 1/20 0.52
KDM4E B2RXH2 1/20 0.47
HPGD P15428 3/20 0.46
LMNA P02545 2/20 0.45
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
PKM P14618 2/20 0.44
HTT P42858 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL676524 0.80 SRC (0.58) SRCL3MBTL1TDP1KDM4EHPGD
SCHEMBL310184 0.80 SRC (0.58) SRCL3MBTL1TDP1KDM4EHPGD
SCHEMBL122230 0.80 SRC (0.58) SRCL3MBTL1TDP1KDM4EHPGD
SCHEMBL259733 0.80 SRC (0.58) SRCL3MBTL1TDP1KDM4EHPGD
SCHEMBL9496224 0.79 TSHR (0.64) HPGDLMNAMEN1KMT2A
SCHEMBL30995990 0.79 SRC (0.64) SRCL3MBTL1TDP1KDM4E
Water SCHEMBL7889250 0.78 SRC (0.56) SRCL3MBTL1TDP1KDM4EHPGD
Hydrochloric Acid SCHEMBL29186320 0.78 SRC (0.56) SRCL3MBTL1TDP1KDM4EHPGD
SCHEMBL5019770 0.78 SRC (0.56) SRCL3MBTL1TDP1KDM4EHPGD
SCHEMBL19212985 0.78 SRC (0.56) SRCL3MBTL1TDP1KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 73 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240228478-A1 COMPOUNDS AND METHODS OF USE TANGO THERAPEUTICS, INC. 2024-07-11 US disclosed
US-20240209017-A1 STING MODULATOR COMPOUNDS, AND METHODS OF MAKING AND USING TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2024-06-27 US disclosed
US-20240067612-A1 PHARMACEUTICAL COMPOSITIONS COMPRISING WRN HELICASE INHIBITORS VIVIDION THERAPEUTICS, INC. 2024-02-29 US disclosed
US-11712715-B2 Surface modification in the vapor phase Quantum-Si Incorporated (US) 2023-08-01 US disclosed
US-11707519-B2 Phosphorylated heptose compounds: process for their preparation and use UNIVERSITY COLLEGE DUBLIN, NATIONAL UNIVERSITY OF IRELAND (IE) 2023-07-25 US disclosed
US-11685761-B2 Cyclic di-nucleotide compounds as sting agonists MERCK SHARP & DOHME LLC (US) 2023-06-27 US disclosed
US-20210139783-A1 FLAME RETARDANT LEVULINIC ACID-BASED COMPOUNDS INTERNATIONAL BUSINESS MACHINES CORPORATION 2021-05-13 US disclosed
US-20190106630-A1 FLAME RETARDANT LEVULINIC ACID-BASED COMPOUNDS INTERNATIONAL BUSINESS MACHINES CORPORATION 2019-04-11 US disclosed
US-20180086784-A1 Phosphonate analogs of HIV inhibitor compounds GILEAD SCIENCES, INC. 2018-03-29 US disclosed
US-9815864-B2 Substituted nucleosides, nucleotides and analogs thereof ALIOS BIOPHARMA, INC. (US) 2017-11-14 US disclosed
US-20070027113-A1 Purine nucleoside phosphorylase inhibitory phosphonate compounds GILEAD SCIENCES, INC. 2007-02-01 US disclosed
US-20070010489-A1 Cellular accumulation of phosphonate analogs of hiv protease inhibitor compounds GILEAD SCIENCES, INC. 2007-01-11 US disclosed
EP-0549073-B1 Novel 2-saccharinylmethyl and 4,5,6,7-tetrahydro-2-saccharinylmethyl phosphates, phosphonates and phosphinates useful as proteolytic enzyme inhibitors and compositions and method of use thereof SANOFI SA (FR) 1997-03-26 EP disclosed
US-5296496-A Treating degenerative diseases STERLING WINTHROP INC. (US) 1994-03-22 US disclosed
EP-0549073-A1 Novel 2-saccharinylmethyl and 4,5,6,7-tetrahydro-2-saccharinylmethyl phosphates, phosphonates and phosphinates useful as proteolytic enzyme inhibitors and compositions and method of use thereof STERLING WINTHROP INC. (US) 1993-06-30 EP disclosed
US-5187173-A Degenerative diseases such as emphysema, rheumatoid arthritis, pancreatitis, cyctic fibrosis and skin disorders STERLING WINTHROP INC. (US) 1993-02-16 US disclosed
US-4301280-A Preparation of 3-substituted cephalosporins LILLY INDUSTRIES LIMITED (GB) 1981-11-17 US disclosed
EP-0019401-A1 Process for preparing enamine derivatives, compounds so produced and process for preparing a 3-hydroxy-cephalosporin Lilly Industries Limited (GB) 1980-11-26 EP disclosed
US-4188382-A Thiazolinyl (thiazolyl) phosphonamidates and phosphoramidates pesticidal and herbicidal compositions based thereon Vsesojuzny Nauchno, et al. (SU) 1980-02-12 US disclosed
US-4113680-A Method for preparing 17 α-ester-21-halo pregnanes TAISHO PHARMACEUTICAL CO., LTD. (JP) 1978-09-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11707519-B2 Phosphorylated heptose compounds: process for their preparation and use PPP6C, G6PD, PFKFB1 SRC 472/4885L3MBTL1 4401/4885TDP1 3328/4885
US-20240209017-A1 STING MODULATOR COMPOUNDS, AND METHODS OF MAKING AND USING STING1, CGAS, MAVS SRC 709/4885L3MBTL1 2681/4885TDP1 78/4885
US-20240067612-A1 PHARMACEUTICAL COMPOSITIONS COMPRISING WRN HELICASE INHIBITORS RECQL, BLM, WRN SRC 3202/4885L3MBTL1 1538/4885TDP1 39/4885
US-20180086784-A1 Phosphonate analogs of HIV inhibitor compounds PIK3CA, TYMP, ITPA SRC 2380/4885L3MBTL1 2435/4885TDP1 1262/4885
US-20240228478-A1 COMPOUNDS AND METHODS OF USE F12, C1R, ABCG2 SRC 3397/4885L3MBTL1 3066/4885TDP1 2792/4885
US-20070010489-A1 Cellular accumulation of phosphonate analogs of hiv protease inhibitor compounds PPA1, PNP, PPME1 SRC 3385/4885L3MBTL1 837/4885TDP1 607/4885
US-11685761-B2 Cyclic di-nucleotide compounds as sting agonists STING1, CGAS, IFNAR1 SRC 4806/4885L3MBTL1 1863/4885TDP1 92/4885
US-20070027113-A1 Purine nucleoside phosphorylase inhibitory phosphonate compounds PNP, TYMP, MTAP SRC 3085/4885L3MBTL1 3935/4885TDP1 237/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.