SCHEMBL4074093

SCHEMBL4074093

CCOP(=O)(Cc1ccc(NC(=O)CCC(=O)NC2CCC(Cc3ccc(Cl)cc3)(N(C)C)CC2)cc1)OCC

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
LMNA P02545 2/20 0.37
ENTPD1 P49961 1/20 0.37
HPGD P15428 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.35
ALDH1A1 P00352 1/20 0.35
MAPT P10636 1/20 0.35
POLB P06746 1/20 0.35
TP53 P04637 1/20 0.35
GAA P10253 2/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
ENPP2 Q13822 4/20 0.35
ATF4 P18848 1/20 0.35
DGAT2 Q96PD7 1/20 0.35
EPHX2 P34913 1/20 0.35
TMEM97 Q5BJF2 1/20 0.35
SIGMAR1 Q99720 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
F10 P00742 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4081068 0.91 THRB (0.39) MEN1KMT2AENTPD1HPGDALDH1A1
SCHEMBL206649 0.88 ENPP2 (0.44) MEN1KMT2ALMNAHPGDSMN1; SMN2
SCHEMBL4074159 0.87 SSTR4 (0.39) MEN1KMT2AENTPD1SMN1; SMN2ALDH1A1
SCHEMBL207874 0.84 KMT2A (0.55) MEN1KMT2ALMNAHPGDSMN1; SMN2
SCHEMBL5160624 0.84 LMNA (0.43) MEN1KMT2ALMNAHPGDSMN1; SMN2
SCHEMBL207100 0.81 NPSR1 (0.43) MEN1KMT2ALMNAHPGDSMN1; SMN2
Butane SCHEMBL4074088 0.80 MEN1 (0.38) MEN1KMT2ALMNAHPGDSMN1; SMN2
SCHEMBL205569 0.79 ENPP2 (0.46) MEN1KMT2AHPGDALDH1A1ENPP2
SCHEMBL206987 0.79 POLB (0.56) MEN1KMT2ALMNAHPGDMAPT
SCHEMBL206932 0.78 LMNA (0.46) MEN1KMT2ALMNAHPGDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1745010-B1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES GRUENENTHAL GMBH (DE) 2009-08-05 EP claimed
EP-1745010-B1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES GRUENENTHAL GMBH (DE) 2009-08-05 EP disclosed