SCHEMBL4074159

SCHEMBL4074159

CCOP(=O)(Cc1ccc(NC(=O)CCC(=O)NC2CCC(Cc3cccc(C)c3)(N(C)C)CC2)cc1)OCC

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SSTR4 P31391 2/20 0.39
SSTR1 P30872 1/20 0.39
KMT2A Q03164 7/20 0.36
TSHR P16473 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
MEN1 O00255 4/20 0.35
HDAC1 Q13547 2/20 0.35
HDAC6 Q9UBN7 1/20 0.35
ALDH1A1 P00352 2/20 0.35
MAPT P10636 2/20 0.35
ENTPD1 P49961 1/20 0.35
NPC1 O15118 1/20 0.35
MAPK1 P28482 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
HDAC2 Q92769 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
LTA4H P09960 1/20 0.34
EPHX2 P34913 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4081068 0.91 THRB (0.39) SSTR4SSTR1KMT2ATSHRMEN1
SCHEMBL206628 0.89 SSTR4 (0.42) SSTR4SSTR1KMT2ATSHRNPSR1
SCHEMBL4074093 0.87 MEN1 (0.38) KMT2ANPSR1MEN1ALDH1A1MAPT
SCHEMBL209344 0.84 ALDH1A1 (0.42) SSTR4SSTR1KMT2AMEN1ALDH1A1
SCHEMBL5161290 0.84 SSTR4 (0.42) SSTR4SSTR1KMT2ATSHRNPSR1
Butane SCHEMBL4074157 0.82 SSTR4 (0.40) SSTR4SSTR1KMT2ATSHRNPSR1
SCHEMBL205569 0.80 ENPP2 (0.46) SSTR4SSTR1KMT2ATSHRMEN1
SCHEMBL204623 0.77 KMT2A (0.48) SSTR4SSTR1KMT2ATSHRNPSR1
SCHEMBL5157976 0.76 SSTR4 (0.45) SSTR4SSTR1KMT2ATSHRNPSR1
SCHEMBL206665 0.76 SSTR4 (0.45) SSTR4SSTR1KMT2ATSHRNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1745010-B1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES GRUENENTHAL GMBH (DE) 2009-08-05 EP claimed
EP-1745010-B1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES GRUENENTHAL GMBH (DE) 2009-08-05 EP disclosed