SCHEMBL4081068

SCHEMBL4081068

CCOP(=O)(Cc1ccc(NC(=O)CCC(=O)NC2CCC(Cc3cccc(Cl)c3)(N(C)C)CC2)cc1)OCC

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.39
HPGD P15428 1/20 0.39
EPHX2 P34913 1/20 0.39
ENPP2 Q13822 1/20 0.38
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
TSHR P16473 1/20 0.36
FSHR P23945 1/20 0.36
IDO1 P14902 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC2 Q92769 1/20 0.36
SIGMAR1 Q99720 3/20 0.35
CACNA1G O43497 1/20 0.35
HSD17B10 Q99714 1/20 0.35
SSTR1 P30872 1/20 0.35
SSTR4 P31391 1/20 0.35
BTK Q06187 1/20 0.35
ALDH1A1 P00352 2/20 0.35
ENTPD1 P49961 1/20 0.35
RORC P51449 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4074159 0.91 SSTR4 (0.39) EPHX2MEN1KMT2ATSHRHDAC1
SCHEMBL4074093 0.91 MEN1 (0.38) HPGDEPHX2ENPP2MEN1KMT2A
SCHEMBL205569 0.89 ENPP2 (0.46) THRBHPGDEPHX2ENPP2MEN1
SCHEMBL5157752 0.84 EPHX2 (0.44) THRBHPGDEPHX2MEN1KMT2A
Butane SCHEMBL4081062 0.82 SIGMAR1 (0.39) THRBHPGDEPHX2MEN1KMT2A
SCHEMBL206628 0.80 SSTR4 (0.42) HPGDENPP2MEN1KMT2ATSHR
SCHEMBL206649 0.80 ENPP2 (0.44) HPGDENPP2MEN1KMT2ASIGMAR1
SCHEMBL206966 0.79 EPHX2 (0.62) THRBHPGDEPHX2MEN1KMT2A
SCHEMBL207303 0.77 SIGMAR1 (0.46) THRBHPGDEPHX2MEN1KMT2A
SCHEMBL206620 0.77 EPHX2 (0.46) THRBHPGDEPHX2SIGMAR1SSTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1745010-B1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES GRUENENTHAL GMBH (DE) 2009-08-05 EP claimed
EP-1745010-B1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES GRUENENTHAL GMBH (DE) 2009-08-05 EP disclosed