SCHEMBL4074654

SCHEMBL4074654

CC(=O)CCc1ccc(-c2ccccc2C(=O)OC(C)(C)C)cc1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.47
ACHE P22303 1/20 0.47
BRS3 P32247 5/20 0.46
SLC6A3 Q01959 3/20 0.43
SLC6A4 P31645 2/20 0.43
LMNA P02545 1/20 0.43
LTB4R2 Q9NPC1 3/20 0.41
NR1H2 P55055 2/20 0.41
NR1H3 Q13133 2/20 0.41
CHRNB2 P17787 1/20 0.40
CHRNB4 P30926 1/20 0.40
CHRNA3 P32297 1/20 0.40
CHRNA4 P43681 1/20 0.40
PTGS2 P35354 1/20 0.40
HCAR2 Q8TDS4 1/20 0.39
FFAR1 O14842 1/20 0.39
FFAR4 Q5NUL3 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3515660 0.85 NR1H2 (0.52) ACHEBRS3SLC6A3SLC6A4LTB4R2
SCHEMBL9854183 0.85 ACHE (0.48) ACHEBRS3SLC6A3SLC6A4LTB4R2
SCHEMBL283 0.85 SLC6A3 (0.48) ALDH1A1ACHEBRS3SLC6A3SLC6A4
SCHEMBL8875151 0.85 ACHE (0.48) ALDH1A1ACHEBRS3SLC6A3SLC6A4
SCHEMBL6983827 0.83 ACHE (0.46) ACHEBRS3SLC6A3SLC6A4LTB4R2
SCHEMBL489306 0.82 NR1H2 (0.48) ACHEBRS3SLC6A3SLC6A4LTB4R2
SCHEMBL4080196 0.82 BRS3 (0.47) ACHEBRS3SLC6A3SLC6A4LTB4R2
SCHEMBL9447390 0.80 ACHE (0.46) ACHEBRS3SLC6A3SLC6A4LTB4R2
SCHEMBL29389473 0.80 BCAT2 (0.52) ALDH1A1SLC6A3SLC6A4LMNACHRNB2
SCHEMBL9531321 0.80 BCAT2 (0.52) ALDH1A1SLC6A3SLC6A4LMNACHRNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2083822-A2 SUBSTITUTED IMIDAZOLES AS BOMBESIN RECEPTOR SUBTYPE-3 MODULATORS Merck & Co., Inc. (US) 2009-08-05 EP disclosed
WO-2008051404-A2 SUBSTITUTED IMIDAZOLES AS BOMBESIN RECEPTOR SUBTYPE-3 MODULATORS MERCK & CO., INC. (US) 2008-05-02 WO disclosed