SCHEMBL4080196

SCHEMBL4080196

CC(O)CCc1ccc(-c2ccccc2C(=O)OC(C)(C)C)cc1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
BRS3 P32247 9/20 0.47
ACHE P22303 1/20 0.46
SLC6A3 Q01959 3/20 0.41
SLC6A4 P31645 2/20 0.41
SCN1A P35498 1/20 0.40
SCN2A Q99250 1/20 0.40
SCN3A Q9NY46 1/20 0.40
KCNA5 P22460 1/20 0.39
LTB4R2 Q9NPC1 2/20 0.39
MMP2 P08253 1/20 0.38
MMP9 P14780 1/20 0.38
MMP12 P39900 1/20 0.38
MMP13 P45452 1/20 0.38
MMP14 P50281 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9854183 0.83 ACHE (0.48) BRS3ACHESLC6A3SLC6A4SCN1A
SCHEMBL3515660 0.83 NR1H2 (0.52) BRS3ACHESLC6A3SLC6A4LTB4R2
SCHEMBL8875151 0.83 ACHE (0.48) BRS3ACHESLC6A3SLC6A4SCN1A
SCHEMBL4074654 0.82 ALDH1A1 (0.47) BRS3ACHESLC6A3SLC6A4LTB4R2
SCHEMBL10449002 0.81 BRS3 (0.46) BRS3LTB4R2MMP2MMP9MMP12
SCHEMBL6983827 0.81 ACHE (0.46) BRS3ACHESLC6A3SLC6A4SCN1A
SCHEMBL283 0.80 SLC6A3 (0.48) BRS3ACHESLC6A3SLC6A4SCN1A
SCHEMBL489306 0.80 NR1H2 (0.48) BRS3ACHESLC6A3SLC6A4SCN1A
SCHEMBL502551 0.79 SLC6A3 (0.42) BRS3ACHESLC6A3SLC6A4SCN1A
SCHEMBL9447390 0.78 ACHE (0.46) BRS3ACHESLC6A3SLC6A4SCN1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2083822-A2 SUBSTITUTED IMIDAZOLES AS BOMBESIN RECEPTOR SUBTYPE-3 MODULATORS Merck & Co., Inc. (US) 2009-08-05 EP disclosed
WO-2008051404-A2 SUBSTITUTED IMIDAZOLES AS BOMBESIN RECEPTOR SUBTYPE-3 MODULATORS MERCK & CO., INC. (US) 2008-05-02 WO disclosed