SCHEMBL4075670

SCHEMBL4075670

O=C(CCc1ccccc1)NCc1ccncc1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.73
CYP3A4 P08684 1/20 0.73
CYP2C9 P11712 1/20 0.73
CYP2C19 P33261 1/20 0.73
ALDH1A1 P00352 4/20 0.71
GAA P10253 2/20 0.71
MAPT P10636 1/20 0.71
SMN1; SMN2 Q16637 1/20 0.66
LMNA P02545 1/20 0.65
TDP1 Q9NUW8 2/20 0.64
TRPV1 Q8NER1 2/20 0.64
HPGD P15428 1/20 0.64
ALOX15 P16050 1/20 0.64
L3MBTL1 Q9Y468 1/20 0.62
MEN1 O00255 1/20 0.60
KMT2A Q03164 1/20 0.60
ERCC1 P07992 1/20 0.60
ERCC4 Q92889 1/20 0.60
PAX8 Q06710 1/20 0.58
TSHR P16473 2/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4071835 1.00 CYP1A2 (0.73) CYP1A2CYP3A4CYP2C9CYP2C19ALDH1A1
SCHEMBL1661081 0.90 TRPV1 (0.76) CYP1A2CYP3A4CYP2C9CYP2C19ALDH1A1
SCHEMBL28571160 0.84 ALDH1A1 (0.60) CYP1A2CYP3A4CYP2C9CYP2C19ALDH1A1
SCHEMBL4076886 0.84 LMNA (0.64) CYP1A2CYP3A4CYP2C9CYP2C19ALDH1A1
SCHEMBL4067164 0.84 CYP3A4 (1.00) CYP1A2CYP3A4CYP2C9CYP2C19ALDH1A1
SCHEMBL16610101 0.84 GAA (0.66) ALDH1A1GAAMAPTSMN1; SMN2LMNA
SCHEMBL11613978 0.83 ALDH1A1 (1.00) CYP3A4ALDH1A1GAAMAPTSMN1; SMN2
SCHEMBL3342974 0.83 GAA (0.66) CYP1A2CYP3A4CYP2C9CYP2C19ALDH1A1
SCHEMBL8792470 0.82 ALDH1A1 (0.71) CYP1A2CYP3A4CYP2C9CYP2C19ALDH1A1
SCHEMBL1894742 0.82 TRPV1 (0.82) CYP1A2CYP3A4CYP2C9CYP2C19ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014111113-A1 ACYLGUANIDINES FOR TREATING OSTEOARTHRITIS MERCK PATENT GMBH (DE) 2014-07-24 WO disclosed
EP-1415986-B1 SPIRO ISOBENZOFURANES AS NEUROPEPTIDE Y RECEPTOR ANTAGONISTS BANYU PHARMA CO LTD (JP) 2009-04-08 EP disclosed
US-7205417-B2 Spiro compounds BANYU PHARMACEUTICAL CO., LTD. (JP) 2007-04-17 US disclosed