SCHEMBL4079335

SCHEMBL4079335

COc1ccc(OC)c(CN2CCN(C(=O)CCCC(=O)O)CC2)c1

nearest known ligand 0.67

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.64
KDM4E B2RXH2 8/20 0.60
ALDH1A1 P00352 6/20 0.60
NPSR1 Q6W5P4 1/20 0.60
LMNA P02545 1/20 0.58
RECQL P46063 1/20 0.58
GAA P10253 1/20 0.57
TDP1 Q9NUW8 1/20 0.57
MEN1 O00255 2/20 0.57
KMT2A Q03164 2/20 0.57
SMN1; SMN2 Q16637 1/20 0.56
TP53 P04637 1/20 0.54
POLB P06746 1/20 0.53
TSHR P16473 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4082831 0.88 MTNR1B (0.67) NPC1KDM4EALDH1A1NPSR1LMNA
SCHEMBL4075869 0.79 ALDH1A1 (0.57) KDM4EALDH1A1NPSR1LMNARECQL
SCHEMBL27923788 0.78 ALDH1A1 (0.67) KDM4EALDH1A1GAATDP1MEN1
SCHEMBL207058 0.77 SIGMAR1 (0.55) NPC1KDM4EALDH1A1NPSR1LMNA
SCHEMBL9426828 0.77 MTNR1B (0.64) NPC1KDM4EALDH1A1NPSR1LMNA
SCHEMBL10041822 0.76 NPC1 (0.62) NPC1KDM4EALDH1A1NPSR1LMNA
SCHEMBL12541529 0.76 NPC1 (0.82) NPC1KDM4EALDH1A1LMNARECQL
SCHEMBL207654 0.75 LMNA (0.52) NPC1KDM4EALDH1A1LMNAGAA
SCHEMBL13504051 0.75 MEN1 (0.59) NPC1KDM4EALDH1A1GAATDP1
SCHEMBL4072689 0.75 ALDH1A1 (0.70) KDM4EALDH1A1LMNAGAAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1745010-B1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES GRUENENTHAL GMBH (DE) 2009-08-05 EP claimed
JP-2007536323-A 2007-12-13 JP claimed
US-20070112007-A1 Cyclohexyl-1, 4-diamine compounds GRUENENTHAL GMBH (DE) 2007-05-17 US claimed
EP-1745010-A1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES Grünenthal GmbH (DE) 2007-01-24 EP claimed
WO-2005110974-A1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES Grünenthal GmbH (DE) 2005-11-24 WO claimed
EP-1745010-B1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES GRUENENTHAL GMBH (DE) 2009-08-05 EP disclosed
US-20070112007-A1 Cyclohexyl-1, 4-diamine compounds GRUENENTHAL GMBH (DE) 2007-05-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070112007-A1 Cyclohexyl-1, 4-diamine compounds PKD1, DDC, DPYD NPC1 46/4885KDM4E 462/4885ALDH1A1 158/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.