SCHEMBL4079501

SCHEMBL4079501

NNC(=O)CCCNc1ccc(C(=O)NN)cn1

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HCAR3 P49019 7/20 0.52
HCAR2 Q8TDS4 1/20 0.40
HDAC1 Q13547 1/20 0.39
NNMT P40261 1/20 0.39
EPHX2 P34913 1/20 0.39
MPO P05164 1/20 0.38
CYP3A4 P08684 1/20 0.38
KDM5A P29375 1/20 0.38
BLM P54132 1/20 0.38
GFER P55789 1/20 0.38
PMP22 Q01453 1/20 0.38
HIF1A Q16665 1/20 0.38
ALDH1A1 P00352 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4072414 0.77 MPO (0.47) HDAC1MPOCYP3A4KDM5ABLM
SCHEMBL217496 0.76 NNMT (0.49) HCAR3HCAR2HDAC1NNMTMPO
SCHEMBL31141613 0.74 HDAC1 (0.57) HCAR3HDAC1GFERALDH1A1
SCHEMBL4070958 0.73 HCAR3 (0.63) HCAR3MPOCYP3A4KDM5ABLM
SCHEMBL4081019 0.73 PRSS1 (0.49) HDAC1MPOCYP3A4KDM5ABLM
SCHEMBL15059555 0.72 HCAR3 (0.61) HCAR3HCAR2NNMT
SCHEMBL18511954 0.72 HDAC1 (0.55) HDAC1ALDH1A1
SCHEMBL25212859 0.72 HCAR3 (0.53) HCAR3NNMTMPOCYP3A4KDM5A
SCHEMBL31292064 0.72 HCAR3 (0.73) HCAR3HCAR2
SCHEMBL4079962 0.72 PRSS1 (0.50) HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009155362-A1 SMALL MOLECULE HEMATOPOIETIC GROWTH FACTOR MIMETIC COMPOUNDS AND THEIR USES LIGAND PHARMACEUTICALS INC. (US) 2009-12-23 WO disclosed