SCHEMBL4081019

SCHEMBL4081019

NNC(=O)CCCCNc1ccc(C(=O)NN)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRSS1 P07477 8/20 0.49
HDAC3 O15379 5/20 0.48
HDAC1 Q13547 5/20 0.48
HDAC2 Q92769 4/20 0.48
F2 P00734 2/20 0.47
PRSS2 P07478 2/20 0.47
PRSS3 P35030 2/20 0.47
TMPRSS6 Q8IU80 2/20 0.47
ST14 Q9Y5Y6 2/20 0.47
MPO P05164 1/20 0.46
CYP3A4 P08684 1/20 0.46
KDM5A P29375 1/20 0.46
BLM P54132 1/20 0.46
GFER P55789 1/20 0.46
PMP22 Q01453 1/20 0.46
HIF1A Q16665 1/20 0.46
NCOR2 Q9Y618 1/20 0.46
HDAC6 Q9UBN7 3/20 0.45
OGG1 O15527 1/20 0.44
KDM4E B2RXH2 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4079962 0.98 PRSS1 (0.50) PRSS1HDAC3HDAC1HDAC2F2
SCHEMBL4072414 0.95 MPO (0.47) PRSS1HDAC3HDAC1HDAC2F2
SCHEMBL4071505 0.88 MPO (0.50) PRSS1MPOCYP3A4KDM5ABLM
SCHEMBL11071683 0.81 PLK1 (0.56) PRSS1HDAC3HDAC1HDAC2F2
SCHEMBL10764251 0.80 SCN5A (0.56) PRSS1HDAC3HDAC1HDAC2MPO
SCHEMBL960116 0.80 CYP3A4 (0.52) HDAC3HDAC1HDAC2MPOCYP3A4
SCHEMBL10457154 0.78 L3MBTL1 (0.61) HDAC3HDAC1HDAC2CYP3A4NCOR2
SCHEMBL4079637 0.76 L3MBTL1 (0.68) MPOCYP3A4KDM5ABLMGFER
SCHEMBL2833538 0.73 CA1 (0.62) ALDH1A1
SCHEMBL4079501 0.73 HCAR3 (0.52) HDAC1MPOCYP3A4KDM5ABLM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009155362-A1 SMALL MOLECULE HEMATOPOIETIC GROWTH FACTOR MIMETIC COMPOUNDS AND THEIR USES LIGAND PHARMACEUTICALS INC. (US) 2009-12-23 WO disclosed