SCHEMBL5157752

SCHEMBL5157752

[CH2]c1ccc(NC(=O)CCC(=O)NC2CCC(Cc3cccc(Cl)c3)(N(C)C)CC2)cc1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.44
THRB P10828 1/20 0.44
HPGD P15428 1/20 0.44
SIGMAR1 Q99720 5/20 0.40
CACNA1G O43497 1/20 0.40
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40
KMT2A Q03164 1/20 0.40
TSHR P16473 2/20 0.39
FSHR P23945 2/20 0.39
KCNQ2 O43526 1/20 0.38
SSTR1 P30872 1/20 0.38
SSTR4 P31391 1/20 0.38
OPRM1 P35372 1/20 0.37
OPRL1 P41146 1/20 0.37
TMEM97 Q5BJF2 1/20 0.37
ACKR3 P25106 1/20 0.37
KDM4E B2RXH2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5161290 0.90 SSTR4 (0.42) MEN1ALDH1A1KMT2ATSHRSSTR1
SCHEMBL5160624 0.89 LMNA (0.43) HPGDSIGMAR1CACNA1GMEN1ALDH1A1
SCHEMBL205569 0.88 ENPP2 (0.46) EPHX2THRBHPGDSIGMAR1CACNA1G
SCHEMBL206966 0.85 EPHX2 (0.62) EPHX2THRBHPGDSIGMAR1MEN1
SCHEMBL4081068 0.84 THRB (0.39) EPHX2THRBHPGDSIGMAR1CACNA1G
Butane SCHEMBL4081062 0.83 SIGMAR1 (0.39) EPHX2THRBHPGDSIGMAR1CACNA1G
SCHEMBL206084 0.83 EPHX2 (0.47) EPHX2THRBHPGDSIGMAR1SSTR1
SCHEMBL206772 0.82 EPHX2 (0.47) EPHX2THRBHPGDSIGMAR1ALDH1A1
SCHEMBL205735 0.82 ALDH1A1 (0.55) EPHX2THRBHPGDSIGMAR1MEN1
SCHEMBL206620 0.81 EPHX2 (0.46) EPHX2THRBHPGDSIGMAR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2007536323-A 2007-12-13 JP claimed
EP-1745010-A1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES Grünenthal GmbH (DE) 2007-01-24 EP claimed
WO-2005110974-A1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES Grünenthal GmbH (DE) 2005-11-24 WO claimed