SCHEMBL4081173

SCHEMBL4081173

Cn1ccc(C(=O)Nc2n[nH]c3cc(C(=O)O)oc23)n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 8/20 0.42
NPC1 O15118 7/20 0.42
PKM P14618 1/20 0.42
SMN1; SMN2 Q16637 4/20 0.42
NFKB1 P19838 2/20 0.42
NFKB2 Q00653 2/20 0.42
RELA Q04206 2/20 0.42
HPGD P15428 1/20 0.42
LMNA P02545 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
KMT2A Q03164 4/20 0.41
MEN1 O00255 3/20 0.41
TP53 P04637 1/20 0.41
ROCK1 Q13464 1/20 0.41
ALDH1A1 P00352 2/20 0.36
PRKCB P05771 1/20 0.35
POLB P06746 2/20 0.35
CYP2C19 P33261 1/20 0.35
KDM5A P29375 1/20 0.35
GSK3B P49841 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2905204 0.91 NPC1 (0.41) RAB9ANPC1PKMSMN1; SMN2NFKB1
SCHEMBL4083886 0.84 AURKA (0.44) RAB9ANPC1PKMSMN1; SMN2NFKB1
SCHEMBL4092000 0.80 HPGD (0.43) RAB9ANPC1PKMSMN1; SMN2NFKB1
SCHEMBL4088627 0.80 PRKCB (0.36) ROCK1PRKCBGSK3BDYRK1A
SCHEMBL650566 0.80 AURKA (0.40) RAB9ANPC1PKMSMN1; SMN2NFKB1
SCHEMBL4088628 0.79 RAB9A (0.43) RAB9ANPC1PKMSMN1; SMN2HPGD
SCHEMBL4088564 0.78 MAPT (0.48) RAB9ANPC1PKMSMN1; SMN2NFKB1
SCHEMBL4078387 0.78 MAPK1 (0.48) RAB9ANPC1PKMSMN1; SMN2LMNA
SCHEMBL4081353 0.78 BRAF (0.39) SMN1; SMN2LMNAL3MBTL1ALDH1A1PRKCB
SCHEMBL4083540 0.77 FGFR1 (0.50) RAB9ANPC1KMT2AMEN1ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2058315-A1 1H-Furo[3,2-C]Pyrazoles active as aurora kinase inhibitors Nerviano Medical Sciences S.r.l. (IT) 2009-05-13 EP disclosed