SCHEMBL4081400

SCHEMBL4081400

CN(C)C1(Cc2cccc(Cl)c2)CCC(NC(=O)CCC(=O)N2CCN(C(=O)O)CC2)CC1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 4/20 0.46
EPHX2 P34913 2/20 0.43
ALDH1A1 P00352 3/20 0.43
THRB P10828 1/20 0.43
HPGD P15428 1/20 0.43
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
NPC1 O15118 1/20 0.40
KDM4E B2RXH2 1/20 0.39
TSHR P16473 1/20 0.39
OPRM1 P35372 1/20 0.39
OPRL1 P41146 1/20 0.39
TP53 P04637 1/20 0.39
MAPT P10636 1/20 0.39
ATM Q13315 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL205163 0.91 SIGMAR1 (0.44) SIGMAR1EPHX2ALDH1A1THRBHPGD
SCHEMBL4081492 0.91 HTR1A (0.45) SIGMAR1EPHX2ALDH1A1THRBHPGD
SCHEMBL208174 0.90 SIGMAR1 (0.43) SIGMAR1EPHX2ALDH1A1THRBHPGD
SCHEMBL207761 0.90 ALDH1A1 (0.51) ALDH1A1MEN1KMT2ASMN1; SMN2NPC1
Propionic Acid SCHEMBL4081494 0.88 SIGMAR1 (0.42) SIGMAR1EPHX2ALDH1A1THRBHPGD
SCHEMBL205991 0.87 USP2 (0.52) ALDH1A1HPGDSMN1; SMN2KDM4ETP53
SCHEMBL4072326 0.87 SIGMAR1 (0.49) SIGMAR1MEN1KMT2AATM
SCHEMBL207353 0.87 THRB (0.43) SIGMAR1EPHX2ALDH1A1THRBHPGD
SCHEMBL205919 0.87 CACNA1G (0.51) SIGMAR1ALDH1A1MEN1KMT2ANPC1
SCHEMBL206991 0.86 EPHX2 (0.43) SIGMAR1EPHX2ALDH1A1THRBHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1745010-B1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES GRUENENTHAL GMBH (DE) 2009-08-05 EP claimed