SCHEMBL4082256

SCHEMBL4082256

Cn1nccc1C(=O)Nc1n[nH]c2cc(C(=O)NC(C)(C)c3ccccc3)oc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 1/20 0.44
ALDH1A1 P00352 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
NAMPT P43490 1/20 0.38
NPC1 O15118 4/20 0.37
RAB9A P51151 4/20 0.37
PKM P14618 1/20 0.37
PHGDH O43175 1/20 0.37
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C19 P33261 1/20 0.36
TSHR P16473 1/20 0.36
HSD17B10 Q99714 1/20 0.36
ABL1 P00519 2/20 0.36
BCR P11274 2/20 0.36
AHR P35869 1/20 0.35
MAPK1 P28482 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
EGLN1 Q9GZT9 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL652354 0.94 AURKA (0.41) AURKAALDH1A1SMN1; SMN2NAMPTNPC1
SCHEMBL4078238 0.87 AURKA (0.43) AURKAALDH1A1SMN1; SMN2PHGDHCYP1A2
SCHEMBL4078547 0.87 AURKA (0.46) AURKAALDH1A1SMN1; SMN2NPC1RAB9A
SCHEMBL4088217 0.85 AURKA (0.51) AURKAABL1BCRMAPK1HTT
SCHEMBL4088628 0.84 RAB9A (0.43) ALDH1A1SMN1; SMN2NAMPTNPC1RAB9A
SCHEMBL4086360 0.84 MAPK1 (0.47) AURKASMN1; SMN2NPC1RAB9APKM
SCHEMBL4089328 0.84 AURKA (0.43) AURKANAMPTRAB9ATSHRABL1
SCHEMBL4093240 0.83 AURKA (0.43) AURKAPHGDHABL1BCRMAPK1
SCHEMBL4083886 0.83 AURKA (0.44) AURKASMN1; SMN2NPC1RAB9APKM
SCHEMBL4078785 0.82 AURKA (0.42) AURKAALDH1A1SMN1; SMN2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2058315-A1 1H-Furo[3,2-C]Pyrazoles active as aurora kinase inhibitors Nerviano Medical Sciences S.r.l. (IT) 2009-05-13 EP disclosed