SCHEMBL4082995

SCHEMBL4082995

CCn1c(-c2cc(Cl)ncn2)[c]c2ccccc21

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 1/20 0.36
PTGER4 P35408 3/20 0.35
TP53 P04637 1/20 0.32
IDO1 P14902 1/20 0.32
CDC7 O00311 1/20 0.31
DAPK3 O43293 1/20 0.31
MAP4K4 O95819 1/20 0.31
PIM1 P11309 1/20 0.31
PRKACA P17612 1/20 0.31
FLT3 P36888 1/20 0.31
CDK8 P49336 1/20 0.31
CLK2 P49760 1/20 0.31
GSK3B P49841 1/20 0.31
CDK7 P50613 1/20 0.31
CDK9 P50750 1/20 0.31
PRKX P51817 1/20 0.31
CDK5 Q00535 1/20 0.31
DYRK1A Q13627 1/20 0.31
PKN2 Q16513 1/20 0.31
MINK1 Q8N4C8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4083502 0.82 SLC6A2 (0.33) SLC6A2CDC7DAPK3MAP4K4PIM1
SCHEMBL3990522 0.82 CYP2D6 (0.38) SLC6A2TP53CYP1A2CYP2D6KMT2A
SCHEMBL323754 0.65 ALDH1A1 (0.41) TP53CYP1A2CYP2D6HTTKMT2A
SCHEMBL4436881 0.62 CYP2D6 (0.47) TP53CDC7DAPK3MAP4K4PIM1
SCHEMBL4078343 0.62 SLC6A2 (0.33) SLC6A2CDC7DAPK3MAP4K4PIM1
SCHEMBL19089318 0.61 EGFR (0.55) TP53CDC7DAPK3MAP4K4PIM1
SCHEMBL632053 0.61 ASIC3 (0.59) TP53CDC7DAPK3MAP4K4PIM1
SCHEMBL29392239 0.61 ASIC3 (0.59) TP53CDC7DAPK3MAP4K4PIM1
SCHEMBL2988060 0.60 CLK4 (0.43) TP53CDC7DAPK3MAP4K4PIM1
SCHEMBL4429838 0.59 CYP2D6 (0.44) TP53CDC7DAPK3MAP4K4PIM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009050235-A1 CGRP ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-04-23 WO disclosed