SCHEMBL4088178

SCHEMBL4088178

CN(c1cc(C(=O)O)ccc1C(=O)[AsH2])C1CC1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR3 P49019 2/20 0.36
TDP1 Q9NUW8 1/20 0.36
MYC P01106 1/20 0.35
ALDH1A1 P00352 3/20 0.34
LCK P06239 1/20 0.34
JAK3 P52333 1/20 0.34
PDK1 Q15118 1/20 0.34
PDK2 Q15119 1/20 0.34
PDK3 Q15120 1/20 0.34
PDK4 Q16654 1/20 0.34
KDM4E B2RXH2 3/20 0.34
NEU3 Q9UQ49 1/20 0.34
POLB P06746 2/20 0.33
GAA P10253 2/20 0.33
ACE2 Q9BYF1 1/20 0.33
NR4A1 P22736 1/20 0.33
HSD17B10 Q99714 1/20 0.33
MAPT P10636 2/20 0.33
NPSR1 Q6W5P4 2/20 0.33
CA12 O43570 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2433377 0.85 ALDH1A1 (0.45) HCAR3TDP1MYCALDH1A1LCK
SCHEMBL31535248 0.78 MYC (0.39) MYC
SCHEMBL31535400 0.74 MYC (0.37) MYCALDH1A1MAPTNPSR1
SCHEMBL31535293 0.74 SCN9A (0.39) MYCALDH1A1LCKJAK3MAPT
SCHEMBL20587133 0.72 ALDH1A1 (0.42) HCAR3TDP1ALDH1A1
SCHEMBL31535307 0.70 CA12 (0.43) ALDH1A1GAAMAPTNPSR1CA12
SCHEMBL31535243 0.69 ALDH1A1 (0.40) TDP1MYCALDH1A1KDM4EGAA
SCHEMBL642243 0.69 HCAR3 (0.53) HCAR3TDP1MYCALDH1A1KDM4E
SCHEMBL194970 0.68 ALDH1A1 (0.46) TDP1ALDH1A1KDM4EPOLBGAA
SCHEMBL3973851 0.68 OPRD1 (0.39) HCAR3TDP1ALDH1A1KDM4ENEU3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074120-A1 TROPANE COMPOUNDS Exelixis, Inc. (US) 2009-07-01 EP disclosed
WO-2009055077-A1 TROPANE COMPOUNDS EXELIXIS, INC. (US) 2009-04-30 WO disclosed