SCHEMBL411220

SCHEMBL411220

O=C(O)Cn1c2ccc(Br)cc2c2cc(Br)ccc21

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.56
TSPO P30536 2/20 0.55
GLA P06280 1/20 0.51
DNMT1 P26358 1/20 0.50
AKR1B10 O60218 1/20 0.49
AKR1A1 P14550 1/20 0.49
AKR1B1 P15121 1/20 0.49
MAPT P10636 2/20 0.49
KRAS P01116 1/20 0.48
PTGDR2 Q9Y5Y4 4/20 0.48
DNM1 Q05193 4/20 0.46
SMN1; SMN2 Q16637 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27547403 0.92 KDM4E (0.72) KDM4ETSPOGLADNMT1AKR1B10
SCHEMBL15486750 0.91 PTGDR2 (0.53) KDM4ETSPOAKR1B1PTGDR2
SCHEMBL15486813 0.91 PTGDR2 (0.51) KDM4ETSPOGLADNMT1AKR1B10
SCHEMBL15485966 0.88 PTGDR2 (0.52) KDM4ETSPOGLADNMT1AKR1B10
SCHEMBL15486120 0.87 TSPO (0.45) KDM4ETSPOGLADNMT1AKR1B10
SCHEMBL21027003 0.85 GLA (0.74) KDM4ETSPOGLADNMT1AKR1B10
SCHEMBL15486330 0.84 TSPO (0.43) KDM4ETSPOGLADNMT1AKR1B10
SCHEMBL14689475 0.84 TSPO (0.54) TSPODNMT1MAPTKRASDNM1
SCHEMBL15489577 0.82 KRAS (0.55) TSPODNMT1MAPTKRASDNM1
SCHEMBL13403413 0.82 FABP4 (0.59) KDM4ETSPODNMT1MAPTDNM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 102 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180318255-A1 Pro-Neurogenic Compounds BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM 2018-11-08 US claimed
EP-2925129-A1 PRO-NEUROGENIC COMPOUNDS Board of Regents of the University of Texas System (US) 2015-10-07 EP claimed
WO-2014031125-A1 PRO-NEUROGENIC COMPOUNDS BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2014-02-27 WO claimed
US-20130040977-A1 Pro-Neurogenic Compounds BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM 2013-02-14 US claimed
CN-112521328-A Preparation method of 3-bromocarbazole 中钢集团南京新材料研究院有限公司 2021-03-19 CN disclosed
US-20190218203-A1 Neuroprotective Compounds and Use Thereof UNIVERSITY OF IOWA RESEARCH FOUNDATION (US) 2019-07-18 US disclosed
US-20190135809-A1 Pro-Neurogenic Compounds NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2019-05-09 US disclosed
US-20190135809-A1 Pro-Neurogenic Compounds NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2019-05-09 US disclosed
US-10183011-B2 Anti-depression compounds BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2019-01-22 US disclosed
US-10183011-B2 Anti-depression compounds BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2019-01-22 US disclosed
US-20180318255-A1 Pro-Neurogenic Compounds BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM 2018-11-08 US disclosed
US-20180127367-A1 Pro-Neurogenic Compounds NATIONAL INSTITUTES OF HEALTH - DIRECTOR DEITR 2018-05-10 US disclosed
US-20130040977-A1 Pro-Neurogenic Compounds BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM 2013-02-14 US disclosed
US-20130040977-A1 Pro-Neurogenic Compounds BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM 2013-02-14 US disclosed
US-20120022096-A1 PRO-NEUROGENIC COMPOUNDS BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2012-01-26 US disclosed
US-20120022096-A1 PRO-NEUROGENIC COMPOUNDS BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2012-01-26 US disclosed
US-20120022096-A1 PRO-NEUROGENIC COMPOUNDS BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2012-01-26 US disclosed
WO-2012006419-A2 PRO-NEUROGENIC COMPOUNDS BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2012-01-12 WO disclosed
WO-2012006419-A2 PRO-NEUROGENIC COMPOUNDS BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2012-01-12 WO disclosed
US-20020193369-A1 Antifungal compounds and uses therefor PROTEZ PHARMACEUTICALS INC. 2002-12-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190218203-A1 Neuroprotective Compounds and Use Thereof NLN, GAP43, BDNF KDM4E 4319/4885TSPO 414/4885GLA 2056/4885
US-20120022096-A1 PRO-NEUROGENIC COMPOUNDS BDNF, GAP43, DCX KDM4E 4210/4885TSPO 2470/4885GLA 163/4885
US-20180127367-A1 Pro-Neurogenic Compounds BDNF, GAP43, DCX KDM4E 4210/4885TSPO 2470/4885GLA 163/4885
US-20020193369-A1 Antifungal compounds and uses therefor CYP51A1, ERG28, TPP1 KDM4E 2603/4885TSPO 1327/4885GLA 1962/4885
US-20180318255-A1 Pro-Neurogenic Compounds BDNF, GAP43, DCX KDM4E 4210/4885TSPO 2470/4885GLA 163/4885
US-10183011-B2 Anti-depression compounds BDNF, DCX, GAP43 KDM4E 3990/4885TSPO 2600/4885GLA 140/4885
US-20190135809-A1 Pro-Neurogenic Compounds BDNF, NES, DCX KDM4E 4356/4885TSPO 2302/4885GLA 179/4885
US-20130040977-A1 Pro-Neurogenic Compounds BDNF, GAP43, DCX KDM4E 4210/4885TSPO 2470/4885GLA 163/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.