SCHEMBL411651

SCHEMBL411651

COC(=O)c1ccc(NCC2=CC(=O)C=CC2=O)cc1Cl

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 5/20 0.43
CYP19A1 P11511 1/20 0.41
NOX4 Q9NPH5 1/20 0.41
ALDH1A1 P00352 2/20 0.39
GAA P10253 2/20 0.39
ALOX15 P16050 2/20 0.39
HSD17B10 Q99714 1/20 0.39
P2RX3 P56373 1/20 0.38
SETD7 Q8WTS6 2/20 0.37
MEN1 O00255 2/20 0.37
LMNA P02545 2/20 0.37
KMT2A Q03164 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
ABL1 P00519 1/20 0.37
MAPT P10636 2/20 0.36
HTT P42858 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
HIF1A Q16665 1/20 0.36
CASR P41180 1/20 0.35
PDK2 Q15119 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL412892 0.88 HSP90AA1 (0.38) CYP19A1ALDH1A1GAAALOX15P2RX3
SCHEMBL412798 0.80 CYP19A1 (0.61) CYP19A1ALDH1A1SETD7MEN1LMNA
SCHEMBL14214714 0.77 AVPR2 (0.47) EGFRNOX4ALDH1A1HSD17B10P2RX3
SCHEMBL20073958 0.75 MAPT (0.41) EGFRNOX4ALDH1A1P2RX3MEN1
SCHEMBL18930912 0.74 AVPR2 (0.49) EGFRALDH1A1P2RX3MEN1LMNA
SCHEMBL410105 0.73 NOX4 (0.36) EGFRCYP19A1NOX4ALDH1A1GAA
SCHEMBL411957 0.72 CAMKK2 (0.35) EGFRCYP19A1NOX4ALDH1A1GAA
SCHEMBL2341546 0.72 ABL1 (0.49) ALDH1A1GAAHSD17B10P2RX3MEN1
SCHEMBL722270 0.71 PTGER4 (0.52) EGFRGAAMEN1LMNAKMT2A
SCHEMBL411958 0.71 HSP90AA1 (0.53) CYP19A1ALDH1A1SETD7MEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120021519-A1 EFFICIENT INDUCTION OF PLURIPOTENT STEM CELLS USING SMALL MOLECULE COMPOUNDS PRESIDENTS AND FELLOWS OF HARVARD COLLEGE (US) 2012-01-26 US disclosed
WO-2010033906-A2 EFFICIENT INDUCTION OF PLURIPOTENT STEM CELLS USING SMALL MOLECULE COMPOUNDS PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2010-03-25 WO disclosed