SCHEMBL412236

SCHEMBL412236

O=C1CCCC(C(=S)c2ccc(C(F)(F)F)cc2)C1=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.39
CES1 P23141 2/20 0.39
GSK3B P49841 2/20 0.37
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
HPGD P15428 1/20 0.37
TSHR P16473 1/20 0.37
LMNA P02545 1/20 0.36
HTT P42858 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
GAA P10253 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
SRD5A2 P31213 1/20 0.35
DHODH Q02127 2/20 0.34
GPR6 P46095 1/20 0.34
PTPN1 P18031 1/20 0.34
CYP1A2 P05177 1/20 0.34
KDM2B Q8NHM5 1/20 0.34
POLB P06746 1/20 0.34
ALDH1A1 P00352 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10740705 0.69 MCL1 (0.64) CES2CES1MEN1KMT2AHPGD
SCHEMBL21060836 0.67 PTGS2 (0.41) MEN1KMT2ACYP1A2ALDH1A1
SCHEMBL134765 0.64 MCL1 (0.62) HTTGAACYP1A2POLBALDH1A1
SCHEMBL7029882 0.63 CES2 (0.60) CES2CES1GSK3BMEN1KMT2A
SCHEMBL10919988 0.62 CES2 (0.58) CES2CES1GSK3BMEN1KMT2A
SCHEMBL6826709 0.62 CYP1A2 (0.33) TSHRCYP1A2
SCHEMBL19650840 0.62 HSD11B1 (0.60) CES2CES1MEN1KMT2ALMNA
SCHEMBL1855141 0.62 HSD11B1 (0.60) CES2CES1MEN1KMT2AHPGD
SCHEMBL1835404 0.61 MCL1 (0.36) POLB
SCHEMBL4023293 0.61 HSD11B1 (0.63) CES2CES1GSK3BLMNAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2595954-B1 (4-TRIFLUORMETHYL-3-THIOBENZOYL)CYCLOHEXANEDIONES AND USE THEREOF AS HERBICIDES BAYER IP GMBH (DE) 2016-05-04 EP claimed
CN-103119020-B (4-trifluoromethyl-3-thiobenzoyl) cyclohexanedione and the purposes as weedicide thereof BAYER INTELLECTUAL PROPERTY GMBH (DE) 2015-08-12 CN claimed
US-8563779-B2 (4-trifluoromethyl-3-thiobenzoyl)cyclohexanediones and use thereof as herbicides BAYER CROPSCIENCE AG (DE) 2013-10-22 US claimed
CN-103119020-A (4-trifluormethyl-3-thiobenzoyl) cyclohexanediones and use thereof as herbicides BAYER CROPSCIENCE AG 2013-05-22 CN claimed
US-20120021902-A1 (4-TRIFLUOROMETHYL-3-THIOBENZOYL)CYCLOHEXANEDIONES AND USE THEREOF AS HERBICIDES BAYER CROPSCIENCE AG (DE) 2012-01-26 US claimed
CN-103119020-B (4-trifluoromethyl-3-thiobenzoyl) cyclohexanedione and the purposes as weedicide thereof BAYER INTELLECTUAL PROPERTY GMBH (DE) 2015-08-12 CN disclosed
CN-103119020-B (4-trifluoromethyl-3-thiobenzoyl) cyclohexanedione and the purposes as weedicide thereof BAYER INTELLECTUAL PROPERTY GMBH (DE) 2015-08-12 CN disclosed
CN-103119020-B (4-trifluoromethyl-3-thiobenzoyl) cyclohexanedione and the purposes as weedicide thereof BAYER INTELLECTUAL PROPERTY GMBH (DE) 2015-08-12 CN disclosed
US-8563779-B2 (4-trifluoromethyl-3-thiobenzoyl)cyclohexanediones and use thereof as herbicides BAYER CROPSCIENCE AG (DE) 2013-10-22 US disclosed
US-8563779-B2 (4-trifluoromethyl-3-thiobenzoyl)cyclohexanediones and use thereof as herbicides BAYER CROPSCIENCE AG (DE) 2013-10-22 US disclosed
JP-2013537523-A 2013-10-03 JP disclosed
EP-2595954-A1 (4-TRIFLUORMETHYL-3-THIOBENZOYL)CYCLOHEXANEDIONES AND USE THEREOF AS HERBICIDES Bayer Intellectual Property GmbH (DE) 2013-05-29 EP disclosed
CN-103119020-A (4-trifluormethyl-3-thiobenzoyl) cyclohexanediones and use thereof as herbicides BAYER CROPSCIENCE AG 2013-05-22 CN disclosed
WO-2012010574-A1 (4-TRIFLUORMETHYL-3-THIOBENZOYL)CYCLOHEXANEDIONES AND USE THEREOF AS HERBICIDES BAYER CROPSCIENCE AG (DE) 2012-01-26 WO disclosed
US-20120021902-A1 (4-TRIFLUOROMETHYL-3-THIOBENZOYL)CYCLOHEXANEDIONES AND USE THEREOF AS HERBICIDES BAYER CROPSCIENCE AG (DE) 2012-01-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120021902-A1 (4-TRIFLUOROMETHYL-3-THIOBENZOYL)CYCLOHEXANEDIONES AND USE THEREOF AS HERBICIDES CBR3, DDT, CYP4X1 CES2 316/4885CES1 688/4885GSK3B 2725/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.