Prazosin

Prazosin

SCHEMBL41258

COc1cc2nc(N3CCN(C(=O)c4ccco4)CC3)nc(N)c2cc1OC.[Cl-].[H+]

nearest known ligand 0.96

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ADRA1AADRA1BADRA1D

The experimentally established mechanism targets of Prazosin. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA1B known ✓ P35368 7/20 0.96
ADRA1A known ✓ P35348 6/20 0.96
ADRA1D known ✓ P25100 4/20 0.96
KDM4E B2RXH2 5/20 0.96
GLA P06280 4/20 0.96
GAA P10253 4/20 0.96
ALDH1A1 P00352 4/20 0.96
MAPT P10636 3/20 0.96
HPGD P15428 3/20 0.96
RAB9A P51151 3/20 0.96
LMNA P02545 2/20 0.96
CYP3A4 P08684 2/20 0.96
ADRA2B P18089 2/20 0.96
ADRA2C P18825 2/20 0.96
OPRM1 P35372 2/20 0.96
HSD17B10 Q99714 2/20 0.96
NPC1 O15118 2/20 0.96
MAPK1 P28482 2/20 0.96
MEN1 O00255 1/20 0.96
SLC22A2 O15244 1/20 0.96

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Prazosin SCHEMBL26524 0.98 ADRA1B (1.00) ADRA1BADRA1AKDM4EGLAGAA
Prazosin SCHEMBL29376126 0.98 ADRA1B (1.00) ADRA1BADRA1AKDM4EGLAGAA
Prazosin SCHEMBL611396 0.97 ADRA1B (1.00) ADRA1BADRA1AKDM4EGLAGAA
Prazosin SCHEMBL29908896 0.97 ADRA1B (1.00) ADRA1BADRA1AKDM4EGLAGAA
Prazosin SCHEMBL41257 0.97 ADRA1B (1.00) ADRA1BADRA1AKDM4EGLAGAA
Prazosin SCHEMBL1172954 0.97 ADRA1B (1.00) ADRA1BADRA1AKDM4EGLAGAA
Prazosin SCHEMBL9663302 0.96 KDM4E (1.00) ADRA1BADRA1AKDM4EGLAGAA
Prazosin SCHEMBL11656542 0.96 KDM4E (1.00) ADRA1BADRA1AKDM4EGLAGAA
Prazosin SCHEMBL29157754 0.95 ADRA1A (0.94) ADRA1BADRA1AKDM4EGLAGAA
SCHEMBL7797445 0.94 ADRA1B (0.93) ADRA1BADRA1AKDM4EGLAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 3343 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025131019-A1 COMPOSITIONS AND METHODS FOR INHIBITING EXPRESSION OF INHIBIN SUBUNIT BETA E (INHBE) SHANGHAI ARGO BIOPHARMACEUTICAL CO., LTD. (CN) 2025-06-26 WO claimed
CN-119234815-A Application of prazosin hydrochloride as strigolactone inhibitor 湖南农业大学 2025-01-03 CN claimed
US-20240252528-A1 Methods Of Treating Metabolic Disorders And Cardiovascular Disease With Inhibin Subunit Beta E (INHBE) Inhibitors REGENERON PHARMACEUTICALS, INC. 2024-08-01 US claimed
CN-118169271-A Method for detecting alpha-adrenergic receptor blocker, SSRI and 5-ARIs and application thereof 巴中市产品质量检验检测中心 2024-06-11 CN claimed
EP-3737676-B1 ACETAL COMPOUNDS AND THERAPEUTIC USES THEREOF LIGAND PHARM INC (US) 2024-03-06 EP claimed
EP-4259279-A1 METHODS OF TREATING METABOLIC DISORDERS AND CARDIOVASCULAR DISEASE WITH INHIBIN SUBUNIT BETA E (INHBE) INHIBITORS REGENERON PHARMACEUTICALS, INC. (US) 2023-10-18 EP claimed
CN-116794183-A Qualitative and quantitative determination method for 25 chemical drugs possibly added in auxiliary antihypertensive health food and/or Chinese patent medicine 山西省检验检测中心(山西省标准计量技术研究院) 2023-09-22 CN claimed
US-20230017661-A1 COMPOSITIONS AND MODULAR NANO- AND MICROPARTICLES FOR THE DELIVERY OF VARIOUS AGENTS AND USE THEREOF VERI NANO INC. (US) 2023-01-19 US claimed
US-20220313726-A1 Methods Of Treating Metabolic Disorders And Cardiovascular Disease With Inhibin Subunit Beta E (INHBE) Inhibitors REGENERON PHARMACEUTICALS, INC. 2022-10-06 US claimed
WO-2022132666-A1 METHODS OF TREATING METABOLIC DISORDERS AND CARDIOVASCULAR DISEASE WITH INHIBIN SUBUNIT BETA E (INHBE) INHIBITORS REGENERON PHARMACEUTICALS, INC. (US) 2022-06-23 WO claimed
EP-0222575-B1 PRAZOSIN-PIRBUTEROL COMBINATION FOR BRONCHODILATION PFIZER INC. (US) 1990-12-27 EP claimed
US-4873330-A AZEOTROPIC DISTILLATION OF HYDRATE WITH SELECTED ORGANIC SOLVENTS ORION-YHTYMA OY (FI) 1989-10-10 US claimed
US-4739055-A HYPOTENSIVE AGENTS ORION-YHTYMA OY (FI) 1988-04-19 US claimed
EP-0222575-A1 Prazosin-pirbuterol combination for bronchodilation PFIZER INC. (US) 1987-05-20 EP claimed
US-4601897-A Prazosin-pirbuterol combination for bronchodilation PFIZER INC. (US) 1986-07-22 US claimed
EP-0126684-A2 Drug delivery system utilizing thermosetting gels MERCK & CO. INC. (US) 1984-11-28 EP claimed
US-4478822-A Drug delivery system utilizing thermosetting gels MERCK & CO., INC. (US) 1984-10-23 US claimed
US-4474752-A DIAMINE MODIFIED POLYOXYETHYLENE-POLYOXYPROPYLENE COPOLYMER MERCK & CO., INC. (US) 1984-10-02 US claimed
US-4472380-A CARBOXYALKYL DIPEPTIDE DERIVATIVES MERCK & CO., INC. (US) 1984-09-18 US claimed
US-4361564-A Renoprotective treatments employing vasodilator compounds EDWARDS K DAVID G 1982-11-30 US claimed