SCHEMBL4128255

SCHEMBL4128255

NC(=O)c1ccccc1C(C1CCCOC1)C1CCCOC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 1/20 0.38
TP53 P04637 1/20 0.37
NAMPT P43490 1/20 0.37
PARP1 P09874 4/20 0.36
KDM4E B2RXH2 2/20 0.34
ALDH1A1 P00352 2/20 0.34
MAPT P10636 1/20 0.34
HPGD P15428 1/20 0.34
TSHR P16473 1/20 0.34
HSD17B10 Q99714 1/20 0.34
NPC1 O15118 1/20 0.34
MAPK8 P45983 1/20 0.34
MAPK9 P45984 1/20 0.34
DPP4 P27487 1/20 0.33
DPP8 Q6V1X1 1/20 0.33
DPP9 Q86TI2 1/20 0.33
DPP7 Q9UHL4 1/20 0.33
RPS6KB1 P23443 1/20 0.33
POLB P06746 1/20 0.33
HTT P42858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6170527 0.73 TP53 (0.42) IRAK4TP53KDM4EALDH1A1MAPT
SCHEMBL6072932 0.73 TP53 (0.46) IRAK4TP53PARP1KDM4EALDH1A1
SCHEMBL6171265 0.72 TP53 (0.48) IRAK4TP53PARP1KDM4EALDH1A1
SCHEMBL5598237 0.72 TP53 (0.48) IRAK4TP53PARP1KDM4EALDH1A1
SCHEMBL5598468 0.72 TP53 (0.48) IRAK4TP53PARP1KDM4EALDH1A1
SCHEMBL22123897 0.69 F2RL1 (0.38) IRAK4TP53NAMPTPARP1KDM4E
SCHEMBL798982 0.69 NAMPT (0.51) NAMPTKDM4EALDH1A1MAPTHPGD
SCHEMBL5598341 0.68 TP53 (0.44) IRAK4TP53PARP1KDM4EALDH1A1
Oxirane SCHEMBL15106942 0.67 ALDH1A1 (0.56) IRAK4PARP1KDM4EALDH1A1MAPT
SCHEMBL633935 0.66 ADRA1A (0.44) PARP1KDM4EALDH1A1MAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1675552-A4 PREPERATION OF 1,6-DISUBSTITUTED AZABENZIMIDAZOLES AS KINASE INHIBITORS GLAXO GROUP LTD (GB) 2009-06-03 EP disclosed
EP-1675552-A2 PREPERATION OF 1,6-DISUBSTITUTED AZABENZIMIDAZOLES AS KINASE INHIBITORS GLAXO GROUP LIMITED (GB) 2006-07-05 EP disclosed
WO-2005037197-A2 PREPERATION OF 1,6-DISUBSTITUTED AZABENZIMIDAZOLES AS KINASE INHIBITORS GLAXO GROUP LIMITED (GB) 2005-04-28 WO disclosed