SCHEMBL4138329

SCHEMBL4138329

Cc1cc(Nc2nccc(-c3cccnc3)n2)ccc1S(=O)(=O)Nc1ncccn1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 15/20 0.60
BCR P11274 13/20 0.60
PRKCA P17252 8/20 0.58
EGFR P00533 5/20 0.55
PRKCD Q05655 4/20 0.55
SRC P12931 5/20 0.55
PRKACA P17612 1/20 0.55
PRKACG P22612 1/20 0.55
PRKACB P22694 1/20 0.55
PDGFRA P16234 6/20 0.54
PDGFRB P09619 5/20 0.54
KIT P10721 1/20 0.53
PRKD3 O94806 1/20 0.52
PRKCG P05129 1/20 0.52
PRKCB P05771 1/20 0.52
LCK P06239 1/20 0.52
PRKCH P24723 1/20 0.52
PRKCI P41743 1/20 0.52
ZAP70 P43403 1/20 0.52
PRKCE Q02156 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4151825 0.90 ABL1 (0.52) ABL1BCRPRKCASRCKIT
SCHEMBL4146823 0.85 IKBKB (0.57) ABL1BCRPRKCAKITJAK3
SCHEMBL4154532 0.81 SYK (0.60) SRCZAP70
SCHEMBL4150544 0.81 SYK (0.46) SRCZAP70JAK3
SCHEMBL4159422 0.81 CDK2 (0.42) JAK3
SCHEMBL7471161 0.78 ABL1 (0.68) ABL1BCRPRKCAEGFRPRKCD
SCHEMBL1978735 0.78 ABL1 (0.69) ABL1BCRPRKCAEGFRPRKCD
Hydrochloric Acid SCHEMBL2081770 0.77 ABL1 (0.68) ABL1BCRPRKCAEGFRPRKCD
SCHEMBL4897551 0.76 ABL1 (0.69) ABL1BCRPRKCAEGFRPRKCD
SCHEMBL7476769 0.76 ABL1 (1.00) ABL1BCRPRKCAEGFRPRKCD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090048282-A1 PYRIMIDINE SULFONAMIDE ANALOGS AND THEIR USE AS AGONISTS OF THE WNT-BETA-CATENIN CELLULAR MESSAGING SYSTEM WYETH (US) 2009-02-19 US claimed
US-20090048282-A1 PYRIMIDINE SULFONAMIDE ANALOGS AND THEIR USE AS AGONISTS OF THE WNT-BETA-CATENIN CELLULAR MESSAGING SYSTEM WYETH (US) 2009-02-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090048282-A1 PYRIMIDINE SULFONAMIDE ANALOGS AND THEIR USE AS AGONISTS OF THE WNT-BETA-CATENIN CELLULAR MESSAGING SYSTEM WNT1, CTNNB1, WNT3A ABL1 3340/4885BCR 1159/4885PRKCA 1301/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.