SCHEMBL4151825

SCHEMBL4151825

Cc1cc(Nc2nccc(-c3ccncc3)n2)ccc1S(=O)(=O)Nc1ncccn1

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 4/20 0.52
BCR P11274 4/20 0.52
SRC P12931 1/20 0.52
PRKCA P17252 3/20 0.50
MTOR P42345 5/20 0.48
PIK3CA P42336 5/20 0.48
PIK3CG P48736 5/20 0.48
CDK1 P06493 4/20 0.48
CDK2 P24941 4/20 0.48
JAK2 O60674 4/20 0.48
JAK3 P52333 4/20 0.48
KIT P10721 1/20 0.46
IKBKB O14920 2/20 0.46
SMG1 Q96Q15 2/20 0.45
MAPK8 P45983 1/20 0.45
MAPK10 P53779 1/20 0.45
KMT2A Q03164 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4138329 0.90 ABL1 (0.60) ABL1BCRSRCPRKCAJAK3
SCHEMBL4146823 0.88 IKBKB (0.57) ABL1BCRPRKCAMTORPIK3CA
SCHEMBL4150544 0.84 SYK (0.46) SRCCDK1CDK2JAK2JAK3
SCHEMBL4154532 0.82 SYK (0.60) SRCCDK2
SCHEMBL4159422 0.81 CDK2 (0.42) CDK1CDK2JAK2JAK3MAPK8
SCHEMBL7467627 0.80 ABL1 (0.61) ABL1BCRSRCPRKCAMTOR
Hydrochloric Acid SCHEMBL8541643 0.76 ABL1 (0.63) ABL1BCRSRCPRKCAMTOR
SCHEMBL6027228 0.74 IKBKB (0.66) CDK2IKBKBMAPK8MAPK10KMT2A
SCHEMBL7467324 0.74 ABL1 (0.76) ABL1BCRSRCPRKCAPIK3CA
SCHEMBL5777773 0.74 ABL1 (0.57) ABL1BCRSRCPRKCAJAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090048282-A1 PYRIMIDINE SULFONAMIDE ANALOGS AND THEIR USE AS AGONISTS OF THE WNT-BETA-CATENIN CELLULAR MESSAGING SYSTEM WYETH (US) 2009-02-19 US claimed
US-20090048282-A1 PYRIMIDINE SULFONAMIDE ANALOGS AND THEIR USE AS AGONISTS OF THE WNT-BETA-CATENIN CELLULAR MESSAGING SYSTEM WYETH (US) 2009-02-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090048282-A1 PYRIMIDINE SULFONAMIDE ANALOGS AND THEIR USE AS AGONISTS OF THE WNT-BETA-CATENIN CELLULAR MESSAGING SYSTEM WNT1, CTNNB1, WNT3A ABL1 3340/4885BCR 1159/4885SRC 1155/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.