SCHEMBL4148404

SCHEMBL4148404

C=CCC(C#N)NC(=O)O

nearest known ligand 0.35

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CTSC P53634 4/20 0.35
GRIK1 P39086 2/20 0.32
GRIK2 Q13002 2/20 0.32
CYP2C19 P33261 1/20 0.32
CPA1 P15085 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9435948 0.77 GRIK1 (0.31) GRIK1GRIK2CYP2C19CPA1
SCHEMBL19745183 0.76 GRIK1 (0.30) GRIK1GRIK2
SCHEMBL24260538 0.74 CTSK (0.44)
SCHEMBL7994665 0.72
Bicarbonate SCHEMBL11765656 0.70 GRIK1 (0.36) GRIK1GRIK2CYP2C19CPA1
SCHEMBL10464154 0.70
SCHEMBL15550726 0.69 CTSC (0.33) CTSCGRIK1GRIK2
SCHEMBL4156798 0.69 CYP2C19 (0.38) GRIK1GRIK2CYP2C19CPA1
SCHEMBL22031610 0.68
SCHEMBL22031609 0.68

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090099168-A1 HIV Integrase inhibitors DONGHI MONICA 2009-04-16 US disclosed
US-20070161639-A1 Hiv integrase inhibitors ISTITUTO DI RICHERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI SPA (IT) 2007-07-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070161639-A1 Hiv integrase inhibitors DPYD, DUT, TYMP CTSC 1500/4885GRIK1 1973/4885GRIK2 2078/4885
US-20090099168-A1 HIV Integrase inhibitors DPYD, DUT, QDPR CTSC 1276/4885GRIK1 2404/4885GRIK2 2619/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.