SCHEMBL4156798

SCHEMBL4156798

C=CCC(C#N)CNC(=O)O

nearest known ligand 0.38

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 2/20 0.38
CYP2D6 P10635 1/20 0.38
GRIK1 P39086 2/20 0.31
GRIK2 Q13002 2/20 0.31
TSHR P16473 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
CPA1 P15085 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3117585 0.84 CYP2D6 (0.50) CYP2C19CYP2D6
Bicarbonate SCHEMBL11768566 0.73 GRIK1 (0.32) CYP2C19GRIK1GRIK2CPA1
SCHEMBL3857558 0.72
SCHEMBL7002068 0.72 CYP2D6 (0.42) CYP2C19CYP2D6GRIK1GRIK2TSHR
SCHEMBL5677966 0.70 ABCC4 (0.47) CYP2C19CYP2D6TSHR
SCHEMBL4148404 0.69 CTSC (0.35) CYP2C19GRIK1GRIK2CPA1
SCHEMBL14110494 0.69 CYP2D6 (0.48) CYP2C19CYP2D6
SCHEMBL19548743 0.68 GRIK1 (0.39) CYP2C19CYP2D6GRIK1GRIK2TSHR
SCHEMBL19552436 0.68 GRIK1 (0.39) CYP2C19CYP2D6GRIK1GRIK2TSHR
SCHEMBL2307423 0.68 CYP2D6 (0.44) CYP2C19CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090099168-A1 HIV Integrase inhibitors DONGHI MONICA 2009-04-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090099168-A1 HIV Integrase inhibitors DPYD, DUT, QDPR CYP2C19 815/4885CYP2D6 341/4885GRIK1 2404/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.