SCHEMBL4149587

SCHEMBL4149587

O=C(N[C@@H]1CCN(C(=O)O)C[C@H]1c1ccc(F)cc1)c1ccc(F)c(C(F)(F)F)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 2/20 0.52
TAS1R1 Q7RTX1 2/20 0.52
TAS1R2 Q8TE23 2/20 0.52
HSD11B1 P28845 1/20 0.40
NOTUM Q6P988 1/20 0.39
SPTLC2 O15270 6/20 0.39
SMYD3 Q9H7B4 1/20 0.39
TLR2 O60603 1/20 0.39
TLR1 Q15399 1/20 0.39
SLC6A9 P48067 2/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
SLC9A1 P19634 1/20 0.38
CYP2C19 P33261 1/20 0.38
KCNQ3 O43525 1/20 0.38
KCNQ2 O43526 1/20 0.38
KCNE1 P15382 1/20 0.38
KCNQ1 P51787 1/20 0.38
PPARG P37231 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4149585 1.00 TAS1R3 (0.52) TAS1R3TAS1R1TAS1R2HSD11B1NOTUM
SCHEMBL4148294 0.93 TAS1R3 (0.51) TAS1R3TAS1R1TAS1R2NOTUMSPTLC2
SCHEMBL4148291 0.93 TAS1R3 (0.51) TAS1R3TAS1R1TAS1R2NOTUMSPTLC2
SCHEMBL4149002 0.90 HSD11B1 (0.52) TAS1R3TAS1R1TAS1R2HSD11B1NOTUM
SCHEMBL4148999 0.90 HSD11B1 (0.52) TAS1R3TAS1R1TAS1R2HSD11B1NOTUM
SCHEMBL13801627 0.87 TAS1R3 (0.52) TAS1R3TAS1R1TAS1R2KMT2A
SCHEMBL13814680 0.87 TAS1R3 (0.52) TAS1R3TAS1R1TAS1R2KMT2A
SCHEMBL4153631 0.85 SPTLC2 (0.44) TAS1R3TAS1R1TAS1R2HSD11B1NOTUM
SCHEMBL4153629 0.85 SPTLC2 (0.44) TAS1R3TAS1R1TAS1R2HSD11B1NOTUM
SCHEMBL4141820 0.85 KCNH2 (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8470816-B2 Nitrogen-containing heterocyclic compound and use thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-06-25 US disclosed
US-20090156572-A1 Nitrogen-containing heterocyclic compound and use thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED 2009-06-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090156572-A1 Nitrogen-containing heterocyclic compound and use thereof NTSR2, NTSR1, HNMT TAS1R3 1426/4885TAS1R1 1216/4885TAS1R2 1033/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.