SCHEMBL4151828

SCHEMBL4151828

[O-][n+]1c(-c2ccccc2)cccc1-c1ccc(C(F)(F)F)cc1

nearest known ligand 0.63

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 5/20 0.63
BACE1 P56817 2/20 0.49
ALDH1A1 P00352 1/20 0.48
TSHR P16473 1/20 0.48
SCN2A Q99250 2/20 0.42
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
TRPV6 Q9H1D0 1/20 0.40
GLO1 Q04760 1/20 0.40
AGXT P21549 1/20 0.39
PTPN5 P54829 1/20 0.39
DPP4 P27487 1/20 0.38
MAPK13 O15264 1/20 0.38
RAF1 P04049 1/20 0.38
MAPK12 P53778 1/20 0.38
MAPK11 Q15759 1/20 0.38
MAPK14 Q16539 1/20 0.38
DHODH Q02127 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4144064 0.81 ALDH1A1 (0.44) ALDH1A1MEN1KMT2A
SCHEMBL14164170 0.79 KIF11 (0.50) KIF11BACE1ALDH1A1TSHRSCN2A
SCHEMBL163728 0.79 KIF11 (1.00) KIF11BACE1ALDH1A1TSHRSCN2A
Water SCHEMBL7382449 0.77 KIF11 (0.95) KIF11BACE1ALDH1A1TSHRSCN2A
Ammonia Solution, Strong SCHEMBL21809401 0.77 KIF11 (0.95) KIF11BACE1ALDH1A1TSHRSCN2A
SCHEMBL27887943 0.77 KIF11 (0.95) KIF11BACE1ALDH1A1TSHRSCN2A
Nitrogen SCHEMBL261370 0.74 KIF11 (0.90) KIF11BACE1ALDH1A1TSHRSCN2A
Hydrazine SCHEMBL27541145 0.74 KIF11 (0.90) KIF11BACE1ALDH1A1TSHRSCN2A
SCHEMBL386142 0.73 ALDH1A1 (0.48) KIF11BACE1ALDH1A1TSHRSCN2A
SCHEMBL11310344 0.73 KIF11 (0.77) KIF11BACE1ALDH1A1TSHRSCN2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8952207-B2 Copper-catalyzed C—H bond arylation THE UNIVERSITY OF HOUSTON SYSTEM (US) 2015-02-10 US disclosed
US-8952207-B2 Copper-catalyzed C—H bond arylation THE UNIVERSITY OF HOUSTON SYSTEM (US) 2015-02-10 US disclosed
US-20090076266-A1 COPPER-CATALYZED C-H BOND ARYLATION THE UNIVERSITY OF HOUSTON SYSTEM (US) 2009-03-19 US disclosed
US-20090076266-A1 COPPER-CATALYZED C-H BOND ARYLATION THE UNIVERSITY OF HOUSTON SYSTEM (US) 2009-03-19 US disclosed
US-20090076266-A1 COPPER-CATALYZED C-H BOND ARYLATION THE UNIVERSITY OF HOUSTON SYSTEM (US) 2009-03-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090076266-A1 COPPER-CATALYZED C-H BOND ARYLATION AOC2, AOC3, DBH KIF11 1251/4885BACE1 2557/4885ALDH1A1 44/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.