SCHEMBL4151852

SCHEMBL4151852

CCc1nc(-c2ccc(Cl)cc2)nc(N2CCCCC2)c1OC(=O)O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.44
ADORA2A P29274 1/20 0.44
ADORA1 P30542 1/20 0.44
TP53 P04637 3/20 0.41
HPGD P15428 2/20 0.41
BCHE P06276 2/20 0.40
ACHE P22303 2/20 0.40
LIPE Q05469 2/20 0.40
MTOR P42345 4/20 0.40
HSD17B10 Q99714 1/20 0.39
MAPT P10636 2/20 0.38
NPC1 O15118 1/20 0.38
TSHR P16473 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
EGLN1 Q9GZT9 2/20 0.38
LMNA P02545 2/20 0.38
ACP1 P24666 1/20 0.38
ALDH1A1 P00352 1/20 0.38
POLB P06746 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4151850 0.83 FABP3 (0.48) ADORA3ADORA2AADORA1TP53HPGD
SCHEMBL8037289 0.80 GABRA2 (0.44) ADORA3ADORA2AADORA1TP53HPGD
SCHEMBL4011569 0.77 PDE4B (0.36) ADORA3ADORA1TP53MAPTTSHR
SCHEMBL4007862 0.76 NAMPT (0.38) ADORA3TP53BCHEACHELIPE
SCHEMBL4011472 0.76 MAPT (0.39) ADORA3HPGDBCHEACHELIPE
SCHEMBL4005144 0.75 PPARA (0.39) ADORA3TP53HSD17B10MAPTNPC1
SCHEMBL4010068 0.72 PPARG (0.40) ADORA3BCHEACHELIPEHSD17B10
SCHEMBL4007708 0.70 CYP1A2 (0.40) ADORA3TP53MAPTRAB9APOLB
SCHEMBL12929476 0.70 MEN1 (0.59) ADORA3ADORA2AADORA1TP53HPGD
SCHEMBL12929363 0.68 MEN1 (0.60) TP53HPGDHSD17B10MAPTNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009080242-A1 SUBSTITUTED 4-AMINOPYRIMIDINE-5-CARBOXYLIC ACID AND USE THEREOF BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2009-07-02 WO disclosed