SCHEMBL4159050

SCHEMBL4159050

C=Cc1cccc(C)c1-c1ncccc1C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.43
NOS3 P29474 1/20 0.42
NOS1 P29475 1/20 0.42
NOS2 P35228 1/20 0.42
PDK2 Q15119 1/20 0.42
METAP2 P50579 1/20 0.40
TGFBR1 P36897 1/20 0.37
PLAU P00749 1/20 0.36
MAPT P10636 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
CNR2 P34972 1/20 0.34
LMNA P02545 1/20 0.33
PDE4A P27815 1/20 0.33
CRHR1 P34998 1/20 0.33
TRPV1 Q8NER1 1/20 0.33
KDM4E B2RXH2 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
TRIM24 O15164 1/20 0.32
TRIM33 Q9UPN9 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27739072 0.88 DPP4 (0.38) CYP2A6NOS3NOS1NOS2PDK2
SCHEMBL12508229 0.85 CYP2A6 (0.46) CYP2A6NOS3NOS1NOS2PDK2
SCHEMBL12320089 0.82 NOS3 (0.54) CYP2A6NOS3NOS1NOS2PDK2
SCHEMBL4151216 0.81 KDM4E (0.43) NOS3NOS1NOS2TGFBR1MAPT
SCHEMBL17696988 0.81 CYP2A6 (0.42) CYP2A6NOS3NOS1NOS2METAP2
SCHEMBL29000603 0.77 CYP2A6 (0.39) CYP2A6NOS3NOS1NOS2METAP2
SCHEMBL24179779 0.76 ALDH1A1 (0.41) CYP2A6MAPTLMNAKDM4ENPC1
SCHEMBL17149986 0.75 CYP2A6 (0.37) CYP2A6NOS3NOS1NOS2METAP2
SCHEMBL20019466 0.74 CYP2A6 (0.41) CYP2A6NOS3NOS1NOS2PDK2
SCHEMBL4150385 0.73 CCR1 (0.48) CYP2A6NOS3NOS1NOS2METAP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8212048-B2 Method of producing aromatic compound SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2012-07-03 US disclosed
US-20090043096-A1 METHOD OF PRODUCING AROMATIC COMPOUND SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2009-02-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090043096-A1 METHOD OF PRODUCING AROMATIC COMPOUND AHR, CYP1A1, ARNT CYP2A6 89/4885NOS3 1302/4885NOS1 756/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.