SCHEMBL4168463

SCHEMBL4168463

O=C1NCCN1c1cccc(CO)c1.OCc1cccc(I)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.46
CYP2C9 P11712 2/20 0.41
CYP2C19 P33261 2/20 0.41
HTR2C P28335 2/20 0.41
HTR1A P08908 2/20 0.41
HTR1D P28221 2/20 0.41
HTR1B P28222 2/20 0.41
HTR2A P28223 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
DRD2 P14416 1/20 0.41
HTR7 P34969 1/20 0.41
DRD3 P35462 1/20 0.41
HTR2B P41595 1/20 0.41
KCNH2 Q12809 1/20 0.41
CFTR P13569 1/20 0.40
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
POLB P06746 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27765009 0.92 ALOX5 (0.52) ALOX5CYP2C9CYP2C19HTR2CHTR1A
SCHEMBL4018203 0.85 ALOX5 (0.47) ALOX5CYP2C9CYP2C19HTR2CHTR1A
SCHEMBL5182221 0.84 FAAH (0.47) ALOX5CYP2C9CYP2C19HTR2CHTR1A
SCHEMBL2885321 0.81 HTR1A (0.48) ALOX5CYP2C9CYP2C19HTR2CHTR1A
SCHEMBL13853418 0.77 CYP2C9 (0.45) ALOX5CYP2C9CYP2C19HTR2CHTR1A
SCHEMBL4013099 0.77 CYP2C9 (0.45) ALOX5CYP2C9CYP2C19HTR2CHTR1A
SCHEMBL2878333 0.77 ITGB3 (0.48) CYP2C9CYP2C19HTR2CHTR1AHTR1D
Hydrochloric Acid SCHEMBL3950851 0.76 CYP2C9 (0.44) ALOX5CYP2C9CYP2C19HTR2CHTR1A
SCHEMBL27765059 0.75 CYP2C9 (0.48) ALOX5CYP2C9CYP2C19HTR2CHTR1A
SCHEMBL7011655 0.75 CYP2C9 (0.43) ALOX5CYP2C9CYP2C19HTR2CHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074098-A2 QUINOLINE COMPOUNDS Wyeth (US) 2009-07-01 EP disclosed
WO-2008049047-A2 QUINOLINE COMPOUNDS WYETH (US) 2008-04-24 WO disclosed