Terbutaline

Terbutaline

SCHEMBL41869

CC(C)(C)NC[C@H](O)c1cc(O)cc(O)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ADRB2

The experimentally established mechanism targets of Terbutaline. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 known ✓ P07550 5/20 1.00
LMNA P02545 5/20 1.00
HIF1A Q16665 4/20 1.00
TSHR P16473 4/20 1.00
KMT2A Q03164 3/20 1.00
CASP7 P55210 2/20 1.00
CYP3A4 P08684 2/20 1.00
CYP2C9 P11712 1/20 1.00
KDM4E B2RXH2 2/20 0.84
MEN1 O00255 2/20 0.84
BLM P54132 2/20 0.84
CASP1 P29466 1/20 0.84
SMN1; SMN2 Q16637 1/20 0.84
ADRA1A P35348 2/20 0.60
ADRB1 P08588 2/20 0.60
HTR1A P08908 1/20 0.60
SLC6A2 P23975 1/20 0.60
SLC6A4 P31645 1/20 0.60
OPRK1 P41145 1/20 0.60
SLC6A3 Q01959 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Terbutaline SCHEMBL4391 1.00 LMNA (1.00) LMNAADRB2HIF1ATSHRKMT2A
Terbutaline SCHEMBL13327959 1.00 LMNA (1.00) LMNAADRB2HIF1ATSHRKMT2A
Terbutaline SCHEMBL404480 0.98 ADRB2 (0.96) LMNAADRB2HIF1ATSHRKMT2A
Terbutaline SCHEMBL11703058 0.98 ADRB2 (0.96) LMNAADRB2HIF1ATSHRKMT2A
Terbutaline SCHEMBL41870 0.92 LMNA (1.00) LMNAADRB2HIF1ATSHRKMT2A
Terbutaline SCHEMBL9614480 0.92 LMNA (1.00) LMNAADRB2HIF1ATSHRKMT2A
Terbutaline SCHEMBL28324621 0.92 LMNA (0.84) LMNAADRB2HIF1ATSHRKMT2A
Terbutaline SCHEMBL26462 0.92 LMNA (1.00) LMNAADRB2HIF1ATSHRKMT2A
Terbutaline SCHEMBL5178614 0.92 LMNA (1.00) LMNAADRB2HIF1ATSHRKMT2A
Terbutaline SCHEMBL3937997 0.92 LMNA (1.00) LMNAADRB2HIF1ATSHRKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 11297 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6423298-B1 None US claimed
EP-4255391-B1 LUMINOL FOR USE IN THE TREATMENT OF SEQUELAE OF A SARS-COV-2 INFECTION METRIOPHARM AG (CH) 2026-05-06 EP claimed
EP-4434588-B1 AEROSOL DELIVERY DEVICE PARI PHARMA GMBH (DE) 2026-04-08 EP claimed
US-20260076872-A1 POLYMER VIALS WITH SUBSTANTIALLY FLAT BOTTOMS AND INJECTION STRETCH BLOW MOLDING METHODS FOR MAKING THE SAME SIO2 MEDICAL PRODUCTS LLC (US) 2026-03-19 US claimed
US-20250242092-A1 SiOx BARRIER FOR PHARMACEUTICAL PACKAGE AND COATING PROCESS SIO2 MEDICAL PRODUCTS INC (US) 2025-07-31 US claimed
CN-120114422-A Atomized inhalation solution for treating bronchial asthma and preparation method and application thereof 中南大学湘雅二医院 2025-06-10 CN claimed
CN-120078752-A Particles for large-dose water-soluble medicine inhalation powder aerosol and preparation method thereof 沈阳药科大学 2025-06-03 CN claimed
CN-119632957-B Terbutaline sulfate solution for aerosol inhalation and preparation method thereof 江苏长泰药业股份有限公司 2025-05-27 CN claimed
EP-4547220-A1 A STABLE ORAL LIQUID COMPOSITION COMPRISING TERBUTALINE & GUAIFENESIN Abdi Ibrahim Ilac Sanayi ve Ticaret Anonim Sirketi (TR) 2025-05-07 EP claimed
US-12257371-B2 SiOx barrier for pharmaceutical package and coating process SIO2 MEDICAL PRODUCTS, LLC (US) 2025-03-25 US claimed
US-4895719-A SUSPENSION, ENCAPSULATION, DRUG DELIVERY LIPOSOME TECHNOLOGY, INC. (US) 1990-01-23 US claimed
EP-0190449-B1 ADDITIVE-CONTAINING PAINTS OECE Industrie Chimiche Spa (IT) 1989-08-09 EP claimed
US-4656027-A ENCAPSULATED DRUGS ASTRA LAKEMEDEL AKTIEBOLAG (SE) 1987-04-07 US claimed
EP-0111144-B1 SUSTAINED RELEASE SOLID DOSAGE FORMS HAVING NON-UNIFORM DISTRIBUTION OF ACTIVE INGREDIENT MERRELL DOW PHARMACEUTICALS INC. (US) 1986-12-03 EP claimed
EP-0189861-A2 Percutaneous absorption accelerator for ionic water-soluble medicine SHOWA DENKO KABUSHIKI KAISHA (JP) 1986-08-06 EP claimed
EP-0069075-B1 PHARMACEUTICAL PREPARATION FOR TREATING GLAUCOMA AND OCULAR HYPERTENSION DISPERSA AG (CH) 1985-11-27 EP claimed
US-4472436-A HIGH DENSITY LIPOOROTEIN, TERBUTALINE NEO-BIONICS, INC. (US) 1984-09-18 US claimed
EP-0043807-B1 1-(DIHYDROXYPHENYL)-2-AMINO-ETHANOL DERIVATIVES; PREPARATION, COMPOSITIONS AND INTERMEDIATES Aktiebolaget Draco (SE) 1984-05-30 EP claimed
EP-0046144-B1 THERAPEUTICALLY ACTIVE DERIVATIVES OF PHENYLETHANOL AMINES Aktiebolaget Draco (SE) 1984-04-11 EP claimed
EP-0069097-A2 Pharmaceutical mixture Astra Läkemedel Aktiebolag (SE) 1983-01-05 EP claimed