SCHEMBL4196595

SCHEMBL4196595

COc1cccc(NC(=O)c2cccc3ccccc23)c1C(=O)NCC1COCCO1

nearest known ligand 0.57

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.57
NPC1 O15118 2/20 0.57
CNR1 P21554 3/20 0.47
CNR2 P34972 3/20 0.47
KMT2A Q03164 4/20 0.45
MEN1 O00255 3/20 0.45
POLB P06746 3/20 0.44
TSHR P16473 1/20 0.43
KDM4E B2RXH2 2/20 0.42
CYP1A2 P05177 1/20 0.42
HPGD P15428 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4192978 0.84 ALDH1A1 (0.49) ALDH1A1NPC1CNR1CNR2KMT2A
SCHEMBL4195582 0.82 POLB (0.47) ALDH1A1NPC1CNR1CNR2KMT2A
SCHEMBL4199022 0.81 CNR1 (0.64) ALDH1A1NPC1CNR1CNR2HPGD
SCHEMBL4200900 0.78 BCL3 (0.61) ALDH1A1POLBTSHRKDM4E
SCHEMBL5223641 0.78 PPARG (0.52) ALDH1A1NPC1KMT2AMEN1POLB
SCHEMBL5225535 0.78 TSHR (0.50) ALDH1A1NPC1CNR1CNR2KMT2A
SCHEMBL5236167 0.77 CNR1 (0.57) ALDH1A1NPC1CNR1CNR2
SCHEMBL4192846 0.76 ALDH1A1 (0.47) ALDH1A1KMT2AMEN1POLBTSHR
SCHEMBL5256886 0.76 TSHR (0.58) ALDH1A1KMT2AMEN1POLBTSHR
SCHEMBL4193276 0.74 ALDH1A1 (0.45) ALDH1A1KMT2AMEN1POLBTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1756044-A1 THERAPEUTIC COMPOUNDS AstraZeneca AB (SE) 2007-02-28 EP claimed
WO-2005115972-A1 THERAPEUTIC COMPOUNDS ASTRAZENECA AB (SE) 2005-12-08 WO claimed
EP-1756044-A1 THERAPEUTIC COMPOUNDS AstraZeneca AB (SE) 2007-02-28 EP disclosed
WO-2005115972-A1 THERAPEUTIC COMPOUNDS ASTRAZENECA AB (SE) 2005-12-08 WO disclosed