SCHEMBL4207201

SCHEMBL4207201

COc1ccc(C2CN(c3ccccc3)CCN2S(=O)(=O)c2cccc3cccnc23)cc1.NC(=O)NC=O

nearest known ligand 0.53

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.53
ALOX15 P16050 2/20 0.53
SMN1; SMN2 Q16637 4/20 0.50
MAPK1 P28482 3/20 0.50
MAPT P10636 3/20 0.50
GAA P10253 5/20 0.47
HTT P42858 2/20 0.47
LMNA P02545 2/20 0.47
HSD17B10 Q99714 1/20 0.47
HSP90AA1 P07900 1/20 0.46
POLB P06746 1/20 0.42
HPGD P15428 1/20 0.42
TP53 P04637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4217064 0.72 FABP1 (0.42) ALDH1A1SMN1; SMN2MAPK1MAPTGAA
SCHEMBL4207423 0.71 GAA (0.45) ALDH1A1MAPK1MAPTGAAHSD17B10
SCHEMBL4208499 0.71 GAA (0.47) ALDH1A1MAPK1MAPTGAAPOLB
SCHEMBL4203707 0.70 ALDH1A1 (0.42) ALDH1A1ALOX15SMN1; SMN2MAPK1MAPT
SCHEMBL4212852 0.69 FABP1 (0.45) ALDH1A1MAPK1MAPTGAAHPGD
SCHEMBL4208204 0.69 ALDH1A1 (0.44) ALDH1A1MAPK1MAPTGAAHTT
SCHEMBL4220008 0.69 ALDH1A1 (0.40) ALDH1A1ALOX15MAPK1MAPTGAA
SCHEMBL1381205 0.69 ALOX15 (0.43) ALDH1A1ALOX15MAPK1MAPTGAA
SCHEMBL4209294 0.67 QPCT (0.42) ALDH1A1MAPK1MAPTGAAHTT
SCHEMBL4037009 0.67 ALDH1A1 (0.52) ALDH1A1ALOX15SMN1; SMN2MAPK1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8404690-B2 Piperazine-2-carboxamide derivatives MERCK SERONO SA (CH) 2013-03-26 US claimed
EP-1592389-B1 PIPERAZINE-2-CARBOXAMIDE DERIVATIVES SERONO LAB (CH) 2009-04-22 EP claimed