SCHEMBL4217064

SCHEMBL4217064

NC(=O)NC=O.O=S(=O)(c1cccc2cccnc12)N1CCN(c2ccccc2-c2ccccc2)CC1Cc1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
FABP1 P07148 5/20 0.42
MAPK1 P28482 3/20 0.42
COMT P21964 1/20 0.40
GAA P10253 3/20 0.40
ALDH1A1 P00352 1/20 0.40
MAPT P10636 2/20 0.39
NPSR1 Q6W5P4 2/20 0.39
HTT P42858 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
USP2 O75604 1/20 0.39
PKM P14618 1/20 0.39
TSHR P16473 1/20 0.38
GFER P55789 1/20 0.38
PKLR P30613 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4212852 0.95 FABP1 (0.45) FABP1MAPK1GAAALDH1A1MAPT
SCHEMBL4208204 0.91 ALDH1A1 (0.44) FABP1MAPK1GAAALDH1A1MAPT
SCHEMBL4214876 0.90 FABP1 (0.40) FABP1MAPK1GAAALDH1A1MAPT
SCHEMBL4208499 0.88 GAA (0.47) FABP1MAPK1GAAALDH1A1MAPT
SCHEMBL4209294 0.85 QPCT (0.42) FABP1MAPK1GAAALDH1A1MAPT
SCHEMBL4220008 0.82 ALDH1A1 (0.40) FABP1MAPK1GAAALDH1A1MAPT
SCHEMBL4207423 0.74 GAA (0.45) FABP1MAPK1GAAALDH1A1MAPT
SCHEMBL4207201 0.72 ALDH1A1 (0.53) MAPK1GAAALDH1A1MAPTHTT
SCHEMBL4038524 0.70 MMP2 (0.34)
SCHEMBL4037792 0.70 ALDH1A1 (0.37) GAAALDH1A1SMN1; SMN2PKMTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8404690-B2 Piperazine-2-carboxamide derivatives MERCK SERONO SA (CH) 2013-03-26 US claimed
EP-1592389-B1 PIPERAZINE-2-CARBOXAMIDE DERIVATIVES SERONO LAB (CH) 2009-04-22 EP claimed