SCHEMBL4221499

SCHEMBL4221499

COC(CCCC(=O)O)(c1ccccc1)c1cncnc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TBXAS1 P24557 8/20 0.42
TBXA2R P21731 7/20 0.42
CYP19A1 P11511 3/20 0.37
HDAC6 Q9UBN7 2/20 0.35
HDAC3 O15379 1/20 0.35
MAPK1 P28482 1/20 0.35
ADRA1A P35348 1/20 0.35
HDAC4 P56524 1/20 0.35
SLC6A3 Q01959 1/20 0.35
HDAC1 Q13547 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
HDAC7 Q8WUI4 1/20 0.35
HDAC2 Q92769 1/20 0.35
HDAC10 Q969S8 1/20 0.35
HDAC11 Q96DB2 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
HDAC9 Q9UKV0 1/20 0.35
HDAC5 Q9UQL6 1/20 0.35
PDK2 Q15119 1/20 0.35
CES1 P23141 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4205855 0.88 TBXAS1 (0.46) TBXAS1TBXA2RHDAC6
SCHEMBL27651289 0.73 KCNN4 (0.46) HDAC6HDAC3MAPK1ADRA1AHDAC4
SCHEMBL5497374 0.69 TBXAS1 (0.49) TBXAS1TBXA2R
SCHEMBL27884300 0.69 HDAC3 (0.48) HDAC6HDAC3MAPK1ADRA1AHDAC4
SCHEMBL2922377 0.69 LMNA (0.45) MAPK1CES1KCNN4
SCHEMBL1051513 0.69 CYP2C19 (0.57) HDAC6HDAC3HDAC4HDAC1SMN1; SMN2
SCHEMBL5753278 0.68 FFAR4 (0.50) HDAC6HDAC3MAPK1ADRA1AHDAC4
SCHEMBL11754754 0.68 CYP2C19 (0.60) HDAC6HDAC3MAPK1ADRA1AHDAC4
SCHEMBL28393601 0.68 ALDH1A1 (0.58) HDAC6HDAC3MAPK1ADRA1AHDAC4
SCHEMBL16468009 0.67 KIF11 (0.55) HDAC6HDAC3MAPK1ADRA1AHDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074093-A2 MATRIX METALLOPROTEINASE INHIBITORS Ranbaxy Laboratories Limited (IN) 2009-07-01 EP claimed
WO-2008023336-A2 MATRIX METALLOPROTEINASE INHIBITORS RANBAXY LABORATORIES LIMITED (IN) 2008-02-28 WO claimed