SCHEMBL4236545

SCHEMBL4236545

CCC(CC)NC(=O)Nc1ccc(Oc2ccc(NC(=O)c3ccc(OC4CCN(CC(C)(C)C(=O)O)CC4)c(CCO)c3)cc2C)cc1F

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 4/20 0.34
ABL1 P00519 3/20 0.33
KIT P10721 3/20 0.33
PKM P14618 1/20 0.33
BRAF P15056 3/20 0.33
KDR P35968 1/20 0.33
DRD2 P14416 1/20 0.33
ADRA1A P35348 1/20 0.33
BCL9 O00512 1/20 0.33
CTNNB1 P35222 1/20 0.33
CSF1R P07333 2/20 0.33
DDR1 Q08345 2/20 0.33
LCK P06239 1/20 0.33
PDGFRB P09619 1/20 0.33
BLK P51451 1/20 0.33
DDR2 Q16832 1/20 0.33
FLT3 P36888 1/20 0.32
ACKR3 P25106 1/20 0.32
DGAT1 O75907 1/20 0.32
RAF1 P04049 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4238724 0.90 MCHR1 (0.37) MCHR1ABL1KITPKMKDR
SCHEMBL4232938 0.87 BCL9 (0.43) BCL9CTNNB1
SCHEMBL4687968 0.84 DRD2 (0.37) MCHR1KITDRD2ADRA1ABCL9
SCHEMBL4228632 0.80 MCHR1 (0.39) MCHR1PKMKDRDRD2TAS1R3
SCHEMBL4228857 0.80 CSF1R (0.38) KITPKMCSF1RPDGFRBFLT3
SCHEMBL4741711 0.78 SSTR5 (0.36) MCHR1KITDRD2ADRA1ABCL9
SCHEMBL4238637 0.78 PKM (0.41) MCHR1PKMBRAFKDRBCL9
SCHEMBL4233470 0.78 MCHR1 (0.40) MCHR1PKMKDRDRD2ADRA1A
SCHEMBL4741716 0.77 CCR5 (0.35) MCHR1ABL1KITDRD2ADRA1A
SCHEMBL4746390 0.77 CSF1R (0.40) MCHR1PKMBRAFKDRBCL9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090233910-A1 Npy antagonists, preparation and uses CEREP (FR) 2009-09-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090233910-A1 Npy antagonists, preparation and uses NPY1R, NPY5R, NPY2R MCHR1 47/4885ABL1 1224/4885KIT 1201/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.