SCHEMBL4245215

SCHEMBL4245215

c1ccc(Nc2nc(-c3n[nH]c4ccccc34)cs2)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 2/20 0.57
SMN1; SMN2 Q16637 6/20 0.52
KMT2A Q03164 6/20 0.51
MAPT P10636 6/20 0.51
MEN1 O00255 5/20 0.51
NFKB1 P19838 3/20 0.51
NFKB2 Q00653 3/20 0.51
RELA Q04206 3/20 0.51
NR1I2 O75469 1/20 0.51
PPP1CA P62136 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51
CSNK2A1 P68400 3/20 0.51
DYRK3 O43781 1/20 0.51
ROCK2 O75116 1/20 0.51
PRKD3 O94806 1/20 0.51
MAP4K4 O95819 1/20 0.51
ROS1 P08922 1/20 0.51
PIM1 P11309 1/20 0.51
RPS6KB1 P23443 1/20 0.51
CDK2 P24941 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1807830 0.77 ALDH1A1 (0.55) SMN1; SMN2KMT2AMAPTMEN1NFKB1
SCHEMBL1822611 0.73 SMN1; SMN2 (0.84) SMN1; SMN2KMT2AMAPTMEN1NFKB1
SCHEMBL7554523 0.73 ALOX5 (0.84) ROCK1SMN1; SMN2KMT2AMAPTMEN1
SCHEMBL15878678 0.73 ROCK1 (1.00) ROCK1SMN1; SMN2KMT2AMAPTMEN1
Bromide SCHEMBL7670429 0.71 ALOX5 (0.82) ROCK1SMN1; SMN2KMT2AMAPTMEN1
Bromide SCHEMBL3354419 0.70 KMT2A (0.58) ROCK1SMN1; SMN2KMT2AMAPTMEN1
SCHEMBL5772080 0.70 KDM4E (0.60) ROCK1SMN1; SMN2KMT2AMAPTMEN1
SCHEMBL28820119 0.70 MAPK10 (0.54) KMT2AMAPTMEN1CDK2GAA
SCHEMBL1886135 0.69 SMN1; SMN2 (1.00) ROCK1SMN1; SMN2KMT2AMAPTMEN1
SCHEMBL12639826 0.68 SMN1; SMN2 (1.00) SMN1; SMN2KMT2AMAPTMEN1NFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009010871-A2 PYRAZOLE DERIVATIVES AS ANTAGONISTS OF ADENOSINE A3 RECEPTOR ADDEX PHARMA S.A. (CH) 2009-01-22 WO disclosed