SCHEMBL4252189

SCHEMBL4252189

COc1cccc(N(F)F)c1

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.50
ENPP2 Q13822 1/20 0.48
CA1 P00915 1/20 0.48
CA2 P00918 1/20 0.48
CA7 P43166 1/20 0.48
CA9 Q16790 1/20 0.48
ALDH1A1 P00352 1/20 0.48
CYP3A4 P08684 1/20 0.48
MTNR1A P48039 6/20 0.45
MTNR1B P49286 6/20 0.45
HSD17B2 P37059 2/20 0.45
ALOX15 P16050 1/20 0.45
HSD17B1 P14061 1/20 0.45
CES2 O00748 1/20 0.44
CES1 P23141 1/20 0.44
NFE2L2 Q16236 1/20 0.43
CHRM5 P08912 1/20 0.42
CA4 P22748 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31256052 0.86 ACHE (0.54) ACHEENPP2CA1CA2CA7
SCHEMBL20979821 0.86 ACHE (0.54) ACHEENPP2CA1CA2CA7
SCHEMBL14163837 0.83 ACHE (0.50) ACHEENPP2CA1CA2CA7
Hydrochloric Acid SCHEMBL28200068 0.82 ALDH1A1 (0.48) ACHEENPP2CA1CA2CA7
SCHEMBL20386564 0.81 CA4 (0.52) ACHEENPP2CA1CA2CA7
SCHEMBL1134073 0.81 CA4 (0.52) ACHEENPP2CA1CA2CA7
SCHEMBL1134082 0.80 MTNR1A (0.61) ACHECA1CA2CA7CA9
SCHEMBL29636366 0.80 ACHE (0.52) ACHECA1CA2CA7CA9
SCHEMBL820669 0.80 ACHE (0.52) ACHECA1CA2CA7CA9
SCHEMBL30054343 0.80 MTNR1A (0.61) ACHECA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107098846-A N- acyl sulfonamides class FBPase inhibitor, its preparation method, pharmaceutical composition and purposes 中国医学科学院药物研究所 2017-08-29 CN disclosed
CN-105384739-A Pyrazolo[3,4-c]pyridine derivative CSPC ZHONGQI PHARMACEUTICAL TECH (SHIJIAZHUANG) CO LTD 2016-03-09 CN disclosed
CN-102126994-B Benzophenone hydrazone derivative and preparation method and application thereof SINOCHEM LANTIAN CO LTD 2014-07-09 CN disclosed
CN-103183623-A A group of benzene sulfonamido benzamide derivatives, and preparation and application thereof INST MEDICINAL BIOTECHNOLOGY 2013-07-03 CN disclosed
CN-101528710-B Aminomethyl-4-imidazoles HOFFMANN LA ROCHE 2012-11-07 CN disclosed
CN-101367815-B Six-membered ring methanamide substituted sulfhydryl pyrrolidine carbpenem compound KBP BIOSCIENCES CO LTD 2012-07-04 CN disclosed
CN-102126994-A Benzophenone hydrazone derivative and preparation method and application thereof SINOCHEM LANTIAN CO LTD 2011-07-20 CN disclosed
CN-101981012-A Novel tetrahydroisoquinoline derivative DAIICHI SANKYO CO LTD 2011-02-23 CN disclosed
CN-101528710-A Aminomethyl-4-imidazoles HOFFMANN LA ROCHE (CH) 2009-09-09 CN disclosed
CN-101367815-A Six-membered ring methanamide substituted sulfhydryl pyrrolidine carbpenem compound SHANDONG XUANZHU MEDICAL SCI T (CN) 2009-02-18 CN disclosed
US-20090036420-A1 BENZAMIDE DERIVATIVES AND THEIR USE FOR TREATING CNS DISORDERS F. HOFFMANN-LA ROCHE AG (CH) 2009-02-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090036420-A1 BENZAMIDE DERIVATIVES AND THEIR USE FOR TREATING CNS DISORDERS GABBR1, GABBR2, CHRM2 ACHE 5/4885ENPP2 1167/4885CA1 1501/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.