SCHEMBL4254583

SCHEMBL4254583

COc1cc(N2C(=O)c3ccc(C)cc3C2=O)ccc1N(C)C

nearest known ligand 0.65

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.52
KMT2A Q03164 3/20 0.52
RAB9A P51151 2/20 0.50
CA9 Q16790 3/20 0.49
CA12 O43570 2/20 0.49
CA1 P00915 2/20 0.49
CA2 P00918 1/20 0.48
ALDH1A1 P00352 3/20 0.47
NPC1 O15118 1/20 0.47
TSHR P16473 1/20 0.47
CASP1 P29466 1/20 0.47
CASP7 P55210 1/20 0.47
HSD17B10 Q99714 1/20 0.47
ESR1 P03372 1/20 0.43
MCHR1 Q99705 1/20 0.42
HTT P42858 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4260752 0.87 ESR1 (0.52) MEN1KMT2AALDH1A1ESR1MCHR1
SCHEMBL4253697 0.87 ALDH1A1 (0.50) MEN1KMT2ARAB9AALDH1A1HSD17B10
SCHEMBL4256269 0.86 NR1H3 (0.52) MEN1KMT2AMCHR1HTT
SCHEMBL4259106 0.86 CYP3A4 (0.43) MEN1KMT2ARAB9AALDH1A1ESR1
SCHEMBL4250037 0.86 CYP3A4 (0.50) MEN1KMT2ARAB9AALDH1A1ESR1
SCHEMBL4253067 0.86 ESR1 (0.52) MEN1KMT2ARAB9AALDH1A1ESR1
SCHEMBL4251879 0.78 NPC1 (0.45) RAB9AALDH1A1NPC1TSHRMCHR1
SCHEMBL4253075 0.78 NPC1 (0.47) MEN1KMT2ARAB9AALDH1A1NPC1
SCHEMBL16602061 0.76 CA9 (0.75) MEN1KMT2ARAB9ACA9CA12
SCHEMBL4256256 0.76 CA9 (0.61) MEN1KMT2ARAB9ACA9CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009054653-A2 ISOINDOLONES WITH HIGH BINDING AFFINITY TO BETA-AMYLOID AGGREGATES AND FIBRILS, AND ITS USE AND PREPARATION METHOD KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2009-04-30 WO claimed
WO-2009054653-A2 ISOINDOLONES WITH HIGH BINDING AFFINITY TO BETA-AMYLOID AGGREGATES AND FIBRILS, AND ITS USE AND PREPARATION METHOD KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2009-04-30 WO disclosed