SCHEMBL4260752

SCHEMBL4260752

COc1ccc2c(c1)C(=O)N(c1ccc(N(C)C)c(OC)c1)C2=O

nearest known ligand 0.58

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 2/20 0.52
MEN1 O00255 7/20 0.52
KMT2A Q03164 7/20 0.52
HTT P42858 1/20 0.50
ALDH1A1 P00352 2/20 0.48
MAPT P10636 1/20 0.48
MCHR1 Q99705 1/20 0.44
GAA P10253 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
NR1H3 Q13133 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4254583 0.87 MEN1 (0.52) ESR1MEN1KMT2AHTTALDH1A1
SCHEMBL4253697 0.87 ALDH1A1 (0.50) ESR1MEN1KMT2AHTTALDH1A1
SCHEMBL4256269 0.86 NR1H3 (0.52) MEN1KMT2AHTTMCHR1NR1H3
SCHEMBL4259106 0.86 CYP3A4 (0.43) ESR1MEN1KMT2AHTTALDH1A1
SCHEMBL4253067 0.86 ESR1 (0.52) ESR1MEN1KMT2AHTTALDH1A1
SCHEMBL4250037 0.86 CYP3A4 (0.50) ESR1MEN1KMT2AHTTALDH1A1
SCHEMBL4258439 0.81 ESR1 (0.61) ESR1MEN1KMT2AHTTALDH1A1
SCHEMBL4254603 0.78 NPC1 (0.51) ESR1MCHR1
SCHEMBL4250774 0.75 NR1H3 (0.56) MEN1KMT2AHTTALDH1A1MCHR1
SCHEMBL4255804 0.75 ESR1 (0.64) ESR1MEN1KMT2AHTTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009054653-A2 ISOINDOLONES WITH HIGH BINDING AFFINITY TO BETA-AMYLOID AGGREGATES AND FIBRILS, AND ITS USE AND PREPARATION METHOD KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2009-04-30 WO claimed
WO-2009054653-A2 ISOINDOLONES WITH HIGH BINDING AFFINITY TO BETA-AMYLOID AGGREGATES AND FIBRILS, AND ITS USE AND PREPARATION METHOD KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2009-04-30 WO disclosed