SCHEMBL4258433

SCHEMBL4258433

CC(C)(C)NCC(O)COc1ccc2c(=O)c(OCc3ccccc3)c(-c3cccc(OCc4ccccc4)c3)oc2c1

nearest known ligand 0.62

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 2/20 0.49
ADRB1 P08588 1/20 0.49
ADRB3 P13945 1/20 0.49
ABCG2 Q9UNQ0 1/20 0.48
CYP2D6 P10635 1/20 0.47
ITGB3 P05106 1/20 0.46
ITGA2B P08514 1/20 0.46
MEN1 O00255 1/20 0.45
RAD52 P43351 1/20 0.45
KMT2A Q03164 1/20 0.45
MAOB P27338 1/20 0.43
PPARG P37231 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4258431 1.00 ADRB2 (0.49) ADRB2ADRB1ADRB3ABCG2CYP2D6
SCHEMBL5320049 0.93 ADRB2 (0.52) ADRB2ADRB1ADRB3ABCG2CYP2D6
SCHEMBL4082991 0.82 PPARG (0.60) ADRB2ADRB1ADRB3CYP2D6ITGB3
SCHEMBL1483979 0.81 ADRB2 (0.52) ADRB2ADRB1ADRB3CYP2D6ITGB3
SCHEMBL1483981 0.81 ADRB2 (0.52) ADRB2ADRB1ADRB3CYP2D6ITGB3
SCHEMBL1483974 0.81 ADRB2 (0.52) ADRB2ADRB1ADRB3CYP2D6ITGB3
SCHEMBL14293136 0.79 ADRB2 (0.49) ADRB2ADRB1ADRB3CYP2D6
SCHEMBL5320651 0.76 MEN1 (0.53) ABCG2CYP2D6MEN1KMT2AMAOB
SCHEMBL4407561 0.76 CYP1A1 (0.48) ADRB2ADRB1ADRB3CYP2D6ITGB3
SCHEMBL20169801 0.76 ABCG2 (0.59) ABCG2MEN1KMT2AMAOBPPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2057137-A1 R-(-) / S-(+)-7-[3-N-SUBSTITUTED AMINO-2-HYDROXYPROPOXY]FLAVONES Council of Scientific and Industrial Research (IN) 2009-05-13 EP disclosed
WO-2008018089-A1 R-(-) / S-(+)-7-[3-N-SUBSTITUTED AMINO-2-HYDROXYPROPOXY] FLAVONES COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2008-02-14 WO disclosed