SCHEMBL4259265

SCHEMBL4259265

CC(C)N1CCN(c2cccc([N+](=O)[O-])c2)C(=O)C1.O=C1CNCCN1c1cccc([N+](=O)[O-])c1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.44
KDM4E B2RXH2 2/20 0.44
TDP1 Q9NUW8 1/20 0.44
MEN1 O00255 2/20 0.40
MAPT P10636 2/20 0.40
KMT2A Q03164 2/20 0.40
HTT P42858 1/20 0.39
HPN P05981 1/20 0.38
HTR1A P08908 1/20 0.38
HTR7 P34969 1/20 0.38
SCN2A Q99250 1/20 0.37
SLC6A2 P23975 1/20 0.36
CHRNB4 P30926 1/20 0.36
CHRNA3 P32297 1/20 0.36
SLC6A3 Q01959 1/20 0.36
BCL2A1 Q16548 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3971995 0.90 ALDH1A1 (0.52) ALDH1A1KDM4ETDP1MEN1MAPT
SCHEMBL3978819 0.87 HPN (0.49) ALDH1A1KDM4EMEN1MAPTKMT2A
SCHEMBL2634714 0.87 HPN (0.49) ALDH1A1KDM4EMEN1MAPTKMT2A
SCHEMBL4256391 0.85 ALDH1A1 (0.47) ALDH1A1KDM4ETDP1MEN1MAPT
SCHEMBL3977939 0.79 ALDH1A1 (0.47) ALDH1A1MEN1MAPTKMT2A
SCHEMBL4079481 0.76 SIRT6 (0.44) ALDH1A1KDM4ETDP1MEN1MAPT
SCHEMBL2634258 0.75 BCL2A1 (0.52) ALDH1A1KDM4EMEN1MAPTKMT2A
SCHEMBL3974009 0.72 DDB1 (0.46) ALDH1A1KDM4EMEN1MAPTKMT2A
SCHEMBL2634327 0.72 MAPT (0.51) ALDH1A1KDM4EMEN1MAPTKMT2A
SCHEMBL4255218 0.72 ALDH1A1 (0.46) ALDH1A1KDM4ETDP1MEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1907385-A4 COMPOUNDS SMITHKLINE BEECHAM CORP (US) 2009-05-06 EP disclosed
EP-1907385-A2 COMPOUNDS SmithKline Beecham Corporation (US) 2008-04-09 EP disclosed
WO-2007018941-A2 PYRIMIDYL-THIOPHENE DERIVATIVES SMITHKLINE BEECHAM CORPORATION (US) 2007-02-15 WO disclosed